SCHEMBL7200542

SCHEMBL7200542

NC(=O)N1CCC(S(=O)(=O)c2ccc(OCc3cccnc3)cc2)C(O)(C(=O)O)C1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 2/20 0.42
RORC P51449 1/20 0.41
MMP13 P45452 6/20 0.40
MMP1 P03956 5/20 0.40
GPR132 Q9UNW8 3/20 0.40
KMT2A Q03164 2/20 0.40
CHRM4 P08173 1/20 0.40
MMP14 P50281 1/20 0.39
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
RAB9A P51151 1/20 0.38
LCK P06239 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7203984 0.90 MMP1 (0.45) ADAMTS4RORCMMP13MMP1MMP14
SCHEMBL7202584 0.89 RORC (0.46) ADAMTS4RORCMMP13MMP1MMP14
SCHEMBL7204248 0.86 MMP1 (0.42) MMP13MMP1MMP14RAB9AMMP3
SCHEMBL7201801 0.84 MMP1 (0.57) ADAMTS4MMP13MMP1
SCHEMBL7201593 0.84 MAOB (0.49) MMP13MMP1MMP14MMP9
SCHEMBL7200563 0.84 MMP1 (0.57) ADAMTS4MMP13MMP1MMP14MMP3
SCHEMBL7201292 0.84 PARP10 (0.44) ADAMTS4RORCMMP13MMP1MMP14
SCHEMBL7205273 0.84 MMP1 (0.56) ADAMTS4MMP13MMP1KMT2AMMP14
SCHEMBL7205347 0.84 MMP1 (0.56) ADAMTS4MMP13MMP1KMT2AMMP14
SCHEMBL7205420 0.84 MMP1 (0.45) ADAMTS4RORCMMP13MMP1MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608104-B2 Antiarthritic agents; anticancer agents PFIZER INC 2003-08-19 US disclosed
US-20020019534-A1 Gem substituted hydroxamic acids PFIZER INC. 2002-02-14 US disclosed
EP-1138680-A1 Gem substituted sulfonyl hydroxamic acids as MMP inhibitors Pfizer Products Inc. (US) 2001-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019534-A1 Gem substituted hydroxamic acids MMP14, TOP2A, ADAMTS1 ADAMTS4 26/4885RORC 2987/4885MMP13 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.