SCHEMBL7201593

SCHEMBL7201593

NC(=O)N1CCC(S(=O)(=O)c2ccc(OCc3cccc(F)c3)cc2)C(O)(C(=O)O)C1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 10/20 0.49
MAOA P21397 7/20 0.49
MMP1 P03956 6/20 0.46
ADAM17 P78536 3/20 0.46
PARP10 Q53GL7 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP14 P50281 1/20 0.46
MMP13 P45452 2/20 0.46
NR4A2 P43354 1/20 0.44
KCNH2 Q12809 1/20 0.44
FAAH O00519 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7203984 0.90 MMP1 (0.45) MMP1ADAM17PARP10MMP2MMP9
SCHEMBL7201801 0.90 MMP1 (0.57) MAOBMMP1ADAM17MMP13
SCHEMBL7200563 0.90 MMP1 (0.57) MAOBMAOAMMP1ADAM17MMP2
SCHEMBL7205420 0.89 MMP1 (0.45) MAOBMMP1ADAM17PARP10MMP2
SCHEMBL7201220 0.89 MMP1 (0.47) MAOBMMP1ADAM17MMP2MMP9
SCHEMBL7207978 0.86 PARP10 (0.45) MMP1PARP10MMP2MMP9MMP14
SCHEMBL7200542 0.84 ADAMTS4 (0.42) MMP1MMP9MMP14MMP13
SCHEMBL7206509 0.84 SCN3A (0.45) MAOBMMP1ADAM17PARP10MMP13
SCHEMBL7205347 0.84 MMP1 (0.56) MMP1ADAM17MMP2MMP9MMP14
SCHEMBL7205273 0.84 MMP1 (0.56) MAOBMMP1ADAM17PARP10MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608104-B2 Antiarthritic agents; anticancer agents PFIZER INC 2003-08-19 US disclosed
US-20020019534-A1 Gem substituted hydroxamic acids PFIZER INC. 2002-02-14 US disclosed
EP-1138680-A1 Gem substituted sulfonyl hydroxamic acids as MMP inhibitors Pfizer Products Inc. (US) 2001-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019534-A1 Gem substituted hydroxamic acids MMP14, TOP2A, ADAMTS1 MAOB 3710/4885MAOA 3573/4885MMP1 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.