SCHEMBL720139

SCHEMBL720139

[c]1cccc2nnc3ccccc3c12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 3/20 0.54
LMNA P02545 3/20 0.35
HTT P42858 2/20 0.35
LCK P06239 1/20 0.35
MAP2K3 P46734 1/20 0.35
MAP2K6 P52564 1/20 0.35
BTK Q06187 1/20 0.35
MAP3K19 Q56UN5 1/20 0.35
NEK10 Q6ZWH5 1/20 0.35
CYP1A2 P05177 3/20 0.34
CYP2C19 P33261 3/20 0.34
KDM4E B2RXH2 6/20 0.33
ALDH1A1 P00352 5/20 0.33
SMN1; SMN2 Q16637 4/20 0.32
MAOA P21397 2/20 0.32
GLA P06280 2/20 0.32
HPGD P15428 2/20 0.32
CASP1 P29466 2/20 0.32
CASP7 P55210 2/20 0.32
HSD17B10 Q99714 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249853 0.76 GPR3 (0.32) GPR3
SCHEMBL2409495 0.73 CYP2A6 (0.33) GPR3CYP1A2ALDH1A1SMN1; SMN2CASP1
Benzonaphthyridine SCHEMBL29600756 0.72 GPR3 (1.00) GPR3LMNAHTTLCKMAP2K3
Benzonaphthyridine SCHEMBL51197 0.72 GPR3 (1.00) GPR3LMNAHTTLCKMAP2K3
Benzonaphthyridine SCHEMBL30897319 0.72 GPR3 (1.00) GPR3LMNAHTTLCKMAP2K3
SCHEMBL4408 0.72 KDM4E (0.57) GPR3LMNACYP1A2KDM4EALDH1A1
SCHEMBL26597 0.72 KDM4E (0.57) GPR3LMNACYP1A2KDM4ESMN1; SMN2
SCHEMBL4824194 0.71 HPRT1 (0.35) CYP1A2ALDH1A1HPGDHSD17B10TDP1
SCHEMBL24104 0.71 HPRT1 (0.35) CYP1A2ALDH1A1HPGDHSD17B10TDP1
SCHEMBL2407351 0.71 HPRT1 (0.35) CYP1A2ALDH1A1HPGDHSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 148 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030216414-A1 Method for preventing tissue injury from hypoxia CELL THERAPEUTICS,INC. 2003-11-20 US claimed
US-6638938-B1 By tissue hypoxia and reoxygenation, comprising administering a compound that inhibits signal transduction by inhibiting cellular accumulation of linoleoyl phosphatidic acid (PA) through an inhibition of the enzyme LPAAT (lysophosphatidic CELL THERAPEUTICS, INC. 2003-10-28 US claimed
EP-0739203-A4 METHOD FOR TREATING DISEASES MEDIATED BY CELLULAR PROLIFERATION IN RESPONSE TO PDGF, EGF, FGF AND VEGF CELL THERAPEUTICS INC (US) 2000-12-20 EP claimed
US-5985926-A VIRICIDES OF AMINE COMPOUNDS AND HYDROCARBONS CELL THERAPEUTICS, INC. (US) 1999-11-16 US claimed
US-5856331-A LYSOPHOSPHATIDIC ACYLTRANSFERASE INHIBITOR CELL THERAPEUTICS, INC. (US) 1999-01-05 US claimed
EP-0739203-A1 METHOD FOR TREATING DISEASES MEDIATED BY CELLULAR PROLIFERATION IN RESPONSE TO PDGF, EGF, FGF AND VEGF CELL THERAPEUTICS, INC. (US) 1996-10-30 EP claimed
EP-0728003-A1 METHOD FOR PREVENTING TISSUE INJURY FROM HYPOXIA CELL THERAPEUTICS, INC. (US) 1996-08-28 EP claimed
EP-0676958-A1 METHOD FOR INHIBITING INTRACELLULAR VIRAL REPLICATION CELL THERAPEUTICS, INC. (US) 1995-10-18 EP claimed
WO-1995019171-A1 METHOD FOR TREATING DISEASES MEDIATED BY CELLULAR PROLIFERATION IN RESPONSE TO PDGF, EGF, FGF AND VEGF CELL THERAPEUTICS, INC. (US) 1995-07-20 WO claimed
WO-1995013075-A1 METHOD FOR PREVENTING TISSUE INJURY FROM HYPOXIA CELL THERAPEUTICS, INC. (US) 1995-05-18 WO claimed
WO-1995012396-A1 METHOD FOR INHIBITING INTRACELLULAR VIRAL REPLICATION CELL THERAPEUTICS, INC. (US) 1995-05-11 WO claimed
CN-117736245-A Organometallic compound, organic light-emitting device, electronic apparatus, and consumer product 三星显示有限公司 2024-03-22 CN disclosed
CN-113766914-B Pentaneamidine analogues and uses thereof 美商奥润沙公司 2024-02-13 CN disclosed
CN-117430589-A 2-aminopyrimidine compound or salt thereof, and preparation method and application thereof 励缔(杭州)医药科技有限公司 2024-01-23 CN disclosed
US-20230233700-A1 METHODS FOR PREPARING ANTIBODY DRUG CONJUGATES GENENTECH, INC. (US) 2023-07-27 US disclosed
EP-0676958-A1 METHOD FOR INHIBITING INTRACELLULAR VIRAL REPLICATION CELL THERAPEUTICS, INC. (US) 1995-10-18 EP disclosed
WO-1995019171-A1 METHOD FOR TREATING DISEASES MEDIATED BY CELLULAR PROLIFERATION IN RESPONSE TO PDGF, EGF, FGF AND VEGF CELL THERAPEUTICS, INC. (US) 1995-07-20 WO disclosed
WO-1995013808-A1 METHOD FOR SELECTIVELY INHIBITING IL-2 SIGNAL TRANSDUCTION CELL THERAPEUTICS, INC. (US) 1995-05-26 WO disclosed
WO-1995013075-A1 METHOD FOR PREVENTING TISSUE INJURY FROM HYPOXIA CELL THERAPEUTICS, INC. (US) 1995-05-18 WO disclosed
WO-1995012396-A1 METHOD FOR INHIBITING INTRACELLULAR VIRAL REPLICATION CELL THERAPEUTICS, INC. (US) 1995-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230233700-A1 METHODS FOR PREPARING ANTIBODY DRUG CONJUGATES FCGRT, MSN, FCGR3B GPR3 4112/4885LMNA 1233/4885HTT 1080/4885
US-20030216414-A1 Method for preventing tissue injury from hypoxia HIF1AN, LPCAT3, PLAAT2 GPR3 2732/4885LMNA 625/4885HTT 4747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.