SCHEMBL7201845

SCHEMBL7201845

COc1ccc2c(c1)C=C(CO)C(c1ccccc1)O2

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.53
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
NFKB1 P19838 3/20 0.43
NFKB2 Q00653 3/20 0.43
RELA Q04206 3/20 0.43
ABCB1 P08183 1/20 0.41
AR P10275 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
CYP19A1 P11511 5/20 0.41
MAOB P27338 1/20 0.39
MTNR1A P48039 1/20 0.39
NR3C1 P04150 2/20 0.39
PGR P06401 1/20 0.39
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7199665 0.87 ALOX5 (0.53) ALOX5PTGS1PTGS2NFKB1NFKB2
SCHEMBL7199661 0.87 ALOX5 (0.50) ALOX5PTGS1PTGS2NFKB1NFKB2
SCHEMBL7203246 0.83 MTNR1A (0.56) ALOX5PTGS1PTGS2NFKB1NFKB2
SCHEMBL7201684 0.79 MTNR1A (0.59) ALOX5PTGS1PTGS2NFKB1NFKB2
SCHEMBL31561627 0.75 NPSR1 (0.60) ALOX5PTGS1PTGS2ABCB1AR
SCHEMBL31561660 0.75 NPSR1 (0.60) ALOX5PTGS1PTGS2ABCB1AR
SCHEMBL7961876 0.74 NFKB1 (0.76) NFKB1NFKB2RELAABCB1NPSR1
Formamide SCHEMBL9730794 0.72 ALOX5 (0.63) ALOX5PTGS1PTGS2
SCHEMBL9030352 0.70 CYP19A1 (0.38) ALOX5PTGS1PTGS2ABCB1AR
SCHEMBL25197813 0.69 NFKB1 (0.54) PTGS1PTGS2NFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602903-B2 Substituted O- and/or S heterocyclic compounds; powerful ligands for melatoninergic receptors. LES LABORATORIES SERVIER (FR) 2003-08-05 US disclosed
US-20020052400-A1 Substituted heterocyclic compounds ADIR ET COMPAGNIE 2002-05-02 US disclosed
US-6313160-B1 FOR THERAPY AND PROPHYLAXIS OF MELATONINERGIC DISORDERS ADIR ET COMPAGNIE (FR) 2001-11-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020052400-A1 Substituted heterocyclic compounds MTNR1A, MTNR1B, CBR1 ALOX5 567/4885PTGS1 570/4885PTGS2 792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.