SCHEMBL7201941

SCHEMBL7201941

CCc1nc2c([nH]1)c(=O)n(CC)c(=O)n2CC(C)C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 0.62
SIRT3 Q9NTG7 2/20 0.62
SIRT5 Q9NXA8 2/20 0.62
PDE5A O76074 4/20 0.56
PDE1A P54750 3/20 0.56
PDE1B Q01064 3/20 0.56
PDE1C Q14123 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
TSHR P16473 2/20 0.56
MEN1 O00255 1/20 0.56
CYP2C19 P33261 1/20 0.56
BLM P54132 1/20 0.56
KMT2A Q03164 1/20 0.56
ADORA2B P29275 7/20 0.53
ADORA2A P29274 6/20 0.53
ADORA1 P30542 4/20 0.53
SIRT2 Q8IXJ6 1/20 0.52
PDE2A O00408 2/20 0.52
ADORA3 P0DMS8 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11069848 0.88 SIRT1 (0.51) SIRT1SIRT3SIRT5PDE5APDE1A
SCHEMBL4623940 0.87 PDE1A (0.55) SIRT1SIRT3SIRT5PDE5APDE1A
SCHEMBL11066985 0.82 SIRT1 (0.54) SIRT1SIRT3SIRT5ADORA2BADORA2A
SCHEMBL7424268 0.80 SIRT1 (0.50) SIRT1SIRT3SIRT5CYP1A2CYP3A4
SCHEMBL11066982 0.80 SIRT1 (0.45) SIRT1SIRT3SIRT5CYP1A2CYP3A4
SCHEMBL7477209 0.77 SIRT1 (0.41) SIRT1SIRT3SIRT5PDE5APDE1A
SCHEMBL4796596 0.77 PDE1A (0.46) SIRT1SIRT3SIRT5PDE5APDE1A
SCHEMBL3399015 0.77 SIRT1 (0.61) SIRT1SIRT3SIRT5CYP1A2CYP3A4
SCHEMBL2917587 0.77 PDE1A (0.78) SIRT1SIRT3SIRT5PDE5APDE1A
SCHEMBL3394252 0.77 SIRT1 (0.61) SIRT1SIRT3SIRT5CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289510-A2 COMPOSITIONS, KITS, AND METHODS FOR PROMOTING DEFINED HEALTH BENEFITS THE PROCTER & GAMBLE COMPANY (US) 2003-03-12 EP disclosed
WO-2001093847-A2 COMPOSITIONS, KITS, AND METHODS FOR PROMOTING DEFINED HEALTH BENEFITS THE PROCTER & GAMBLE COMPANY (US) 2001-12-13 WO disclosed