SCHEMBL7203775

SCHEMBL7203775

O=c1cc(NC2CCNCC2)c2ccccc2n1-c1nc2ccccc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 1/20 0.49
AURKA O14965 9/20 0.48
CHEK1 O14757 6/20 0.44
HTR3A P46098 1/20 0.42
PDGFRB P09619 1/20 0.41
FGFR1 P11362 1/20 0.41
KDR P35968 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OGFRL1 Q5TC84 1/20 0.40
NR4A2 P43354 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7199711 0.88 JAK1 (0.52) JAK1AURKACHEK1
SCHEMBL7204767 0.84 JAK1 (0.56) JAK1AURKAOPRM1OPRK1KCNH2
SCHEMBL5111478 0.79 NR4A2 (0.51) JAK1AURKACHEK1HTR3AOPRM1
SCHEMBL7202162 0.79 AURKA (0.45) AURKAPDGFRBFGFR1KDR
SCHEMBL7201841 0.76 AURKA (0.43) AURKA
SCHEMBL5308810 0.74 AURKA (0.62) AURKAPDGFRBKDR
SCHEMBL7206567 0.74 ACP1 (0.52) AURKA
SCHEMBL7203420 0.72 ALDH1A1 (0.48) AURKA
SCHEMBL7086067 0.72 FLT3 (0.44) PDGFRBFGFR1KDRKCNH2
SCHEMBL7200373 0.71 ACP1 (0.55) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6605617-B2 Treating a patient in need of an inhibitor of vascular endothelial growth factor receptor tyrosine kinase CHIRON CORPORATION 2003-08-12 US disclosed