SCHEMBL7208679

SCHEMBL7208679

NC(=O)c1ccc(C2=NNC=CC=C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 10/20 0.39
MKNK2 Q9HBH9 10/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CYP17A1 P05093 1/20 0.37
ERN1 O75460 1/20 0.36
MAP4K4 O95819 1/20 0.36
IKBKB O14920 2/20 0.36
RIPK1 Q13546 1/20 0.35
CHUK O15111 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
PARP15 Q460N3 1/20 0.35
PARP14 Q460N5 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP16 Q8N5Y8 1/20 0.35
PARP11 Q9NR21 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5155602 0.72 BCAT2 (0.45) MAP4K4ALDH1A1
SCHEMBL3969262 0.70
Hydrochloric Acid SCHEMBL3963502 0.68
SCHEMBL27205294 0.68
SCHEMBL1002578 0.67 CA2 (0.67) MKNK1MKNK2CA12CA1CA2
Terephthalamide SCHEMBL23774 0.65 PARP1 (0.71) CA12CA1CA2CA9CA14
SCHEMBL15748062 0.64 MKNK1 (0.53) MKNK1MKNK2CA12CA1CA2
SCHEMBL28610546 0.64 CA2 (0.56) MKNK1MKNK2CA12CA1CA2
Terephthalamide SCHEMBL11512422 0.62 PARP1 (0.67) CA12CA1CA2CA9CA14
Terephthalamide SCHEMBL7508927 0.62 PARP1 (0.67) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907644-A4 PHARMACEUTICAL PREPARATION MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-0907644-A1 PHARMACEUTICAL PREPARATION Merck & Co., Inc. (US) 1999-04-14 EP disclosed
WO-1998000405-A1 PHARMACEUTICAL PREPARATION MERCK & CO., INC. (US) 1998-01-08 WO disclosed