SCHEMBL7211504

SCHEMBL7211504

COC(=O)[C@H](CN1C(=O)NC2(CCN(C(=O)O)CC2)C1=O)NC(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KYNU Q16719 1/20 0.48
CCR1 P32246 1/20 0.44
ALDH1A1 P00352 2/20 0.44
ALOX15 P16050 1/20 0.44
ITGB3 P05106 2/20 0.42
ITGA2B P08514 2/20 0.42
TGM2 P21980 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.41
CTSK P43235 3/20 0.41
CYP3A4 P08684 2/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
OPRK1 P41145 1/20 0.41
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41
CTSS P25774 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7397329 0.84 KYNU (0.40) KYNUALDH1A1ALOX15CTSKCYP3A4
SCHEMBL7216458 0.81 ITGB3 (0.51) ITGB3ITGA2B
SCHEMBL7211673 0.80 TACR1 (0.41) ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL7211164 0.80 ITGB3 (0.47) ITGB3ITGA2BCTSL
SCHEMBL7211500 0.79 CCR1 (0.41) KYNUCCR1ALDH1A1ITGB3ITGA2B
SCHEMBL20522430 0.74 KYNU (0.54) KYNUCCR1ALDH1A1ALOX15CTSK
SCHEMBL29440261 0.74 KYNU (0.51) KYNUALDH1A1ALOX15CTSKOPRK1
SCHEMBL20522431 0.74 KYNU (0.54) KYNUCCR1ALDH1A1ALOX15CTSK
SCHEMBL6506646 0.72 CASP1 (0.59) KYNUALDH1A1ALOX15CTSKOPRK1
SCHEMBL5651104 0.72 KYNU (0.53) KYNUALDH1A1ALOX15CTSKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620820-B2 Imidazole dione or one, thione derivatives as antitumor and antiinflammatory agents, also treats cardiovascular disease, nephropathies and retinopathies HOECHST AKTIENGESELLSCHAFT (DE) 2003-09-16 US disclosed
US-20020119999-A1 Novel inhibitors of bone reabsorption and antagonists of vitronectin receptors HOECHST AKTIENGESELLSCHAFT 2002-08-29 US disclosed
US-20010021708-A1 Novel inhibitors of bone reabsorption and antagonists of vitronectin receptors WEHNER VOLKMAR (DE) 2001-09-13 US disclosed
US-6218415-B1 THERAPY OF BONE REABSORPTION BY OSTEOCLASTS, TUMOR GROWTH AND TUMOR METASTASIS, INFLAMMATION, CARDIOVASCULAR DISEASE, NEPHROPATHIES AND RETINOPATHIES HOECHST AKTIENGESELLSCHAFT (DE) 2001-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010021708-A1 Novel inhibitors of bone reabsorption and antagonists of vitronectin receptors ADGRF1, CALCR, SOST KYNU 3220/4885CCR1 562/4885ALDH1A1 4551/4885
US-20020119999-A1 Novel inhibitors of bone reabsorption and antagonists of vitronectin receptors ADGRF1, CALCR, SOST KYNU 3220/4885CCR1 562/4885ALDH1A1 4551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.