SCHEMBL7214526

SCHEMBL7214526

NC(=O)[C@@H]1CCN(Cc2csc3c(Cl)ncnc23)C1=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.33
F10 P00742 2/20 0.33
PLG P00747 2/20 0.33
PLAT P00750 2/20 0.33
PROC P04070 2/20 0.33
MAPT P10636 2/20 0.31
RAB9A P51151 1/20 0.31
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6223127 0.88 CSF1R (0.33) MAPTRAB9A
SCHEMBL7214529 0.84 MAPT (0.32) F2F10PLGPLATPROC
Trifluoroacetic Acid SCHEMBL7214364 0.82 L3MBTL1 (0.30)
SCHEMBL7214400 0.82 F10 (0.40) F2F10PLGPLATPROC
SCHEMBL7448311 0.82 F10 (0.40) F2F10PLGPLATPROC
SCHEMBL7219265 0.76 F2 (0.37) F2F10PLGPLATPROC
SCHEMBL7449196 0.76 F2 (0.37) F2F10PLGPLATPROC
SCHEMBL7213490 0.76 F10 (0.40) F2F10PLGPLATPROC
SCHEMBL7456508 0.76 F10 (0.40) F2F10PLGPLATPROC
SCHEMBL7213537 0.72 SELE (0.44) F2F10PLGPLATPROC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602864-B1 Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-08-05 US disclosed
EP-0944386-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
US-6281227-B1 INHIBITORS OF THE ACTIVITY OF FACTOR XA. AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-08-28 US disclosed
WO-2001039759-A2 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-06-07 WO disclosed