SCHEMBL7216469

SCHEMBL7216469

CCOCCOc1ccc(NC(=O)c2c[nH]c3c2-c2nn(C)cc2CCC3)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
AURKA O14965 4/20 0.39
NR3C1 P04150 5/20 0.39
ABCB1 P08183 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
TP53 P04637 2/20 0.38
EPHX2 P34913 1/20 0.38
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 5/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7217055 0.94 NPC1 (0.48) NPC1RAB9AAURKANR3C1ABCB1
SCHEMBL7216803 0.90 NR3C1 (0.41) NPC1RAB9ANR3C1TP53EPHX2
SCHEMBL7216549 0.84 ROCK2 (0.37) NPC1RAB9AAURKANR3C1TP53
SCHEMBL7216265 0.83 NPC1 (0.38) NPC1RAB9AAURKANR3C1TP53
SCHEMBL7217034 0.80 GCK (0.38)
SCHEMBL7222815 0.80 GCK (0.38)
SCHEMBL7216813 0.79 F10 (0.39) NPC1RAB9ATP53
SCHEMBL7216626 0.78 APLNR (0.44) NPC1RAB9ATP53MAPTHPGD
SCHEMBL6831069 0.78 NAMPT (0.53) NPC1RAB9AMAPTHPGDHTT
SCHEMBL7216812 0.77 NPC1 (0.56) NPC1RAB9ATP53MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6653471-B2 Tricyclic heteroaromatic compounds containing pyrrole ring; central nervous system disorder treatment; side effect reduction NEUROGEN CORPORATION 2003-11-25 US disclosed