SCHEMBL7217034

SCHEMBL7217034

Cn1cc2c(n1)-c1c(C(=O)Nc3ccc(O[C@H]4CCOC4)cc3)c[nH]c1CCC2

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCK P35557 1/20 0.38
KCNH2 Q12809 1/20 0.38
DYRK1A Q13627 4/20 0.36
GSK3B P49841 3/20 0.36
DDX3X O00571 1/20 0.35
GRM5 P41594 3/20 0.34
ACACB O00763 2/20 0.34
NAMPT P43490 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7222815 1.00 GCK (0.38) GCKKCNH2DYRK1AGSK3BDDX3X
SCHEMBL7217055 0.82 NPC1 (0.48)
SCHEMBL7216469 0.80 NPC1 (0.42)
SCHEMBL7216549 0.80 ROCK2 (0.37) ACACB
SCHEMBL7216812 0.78 NPC1 (0.56)
SCHEMBL7216626 0.75 APLNR (0.44) NAMPT
SCHEMBL6831069 0.75 NAMPT (0.53) NAMPT
SCHEMBL7216813 0.75 F10 (0.39) KCNH2
SCHEMBL7216265 0.73 NPC1 (0.38) IRAK4
SCHEMBL6834309 0.73 LMNA (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6653471-B2 Tricyclic heteroaromatic compounds containing pyrrole ring; central nervous system disorder treatment; side effect reduction NEUROGEN CORPORATION 2003-11-25 US disclosed