SCHEMBL7216601

SCHEMBL7216601

CCCOCCOc1ccc(Oc2ccc3c(c2)C=C(C(=O)O)CCS3(=O)=O)cc1C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.37
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
WDR5 P61964 3/20 0.32
RXRA P19793 1/20 0.32
PPARD Q03181 5/20 0.32
PPARA Q07869 4/20 0.32
PPARG P37231 3/20 0.32
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
RARA P10276 1/20 0.31
LMNA P02545 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216023 0.91 L3MBTL1 (0.34) RARBHTTMEN1KMT2APPARD
SCHEMBL7222573 0.90 POLB (0.38) RARBMEN1KMT2APPARDKDM4E
SCHEMBL7222487 0.90 RARB (0.38) RARBPPARDPPARAPPARGKDM4E
SCHEMBL7215993 0.87 KMT2A (0.39) RARBKMT2AKDM4EALDH1A1LMNA
SCHEMBL7216344 0.84 THRB (0.34) MEN1KMT2A
SCHEMBL7218340 0.83 LTA4H (0.40) HTTKMT2ALMNAL3MBTL1
SCHEMBL7216783 0.82 PPARD (0.35) RARBMEN1KMT2APPARDPPARG
SCHEMBL7247416 0.82 RARB (0.46) RARBKDM4ERARALMNA
SCHEMBL7218217 0.82 S1PR1 (0.36) MEN1KMT2APPARDPPARAPPARG
SCHEMBL7215961 0.81 HRH3 (0.39) RARBKMT2ARXRAPPARGKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed