SCHEMBL7218902

SCHEMBL7218902

CO/N=C1/C[C@@H](C(=O)NCc2ccc(OC)c(OC)c2)N(C(=O)C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 6/20 0.50
OXTR P30559 2/20 0.50
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
AGTR1 P30556 2/20 0.47
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
POLB P06746 1/20 0.46
AVPR1A P37288 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4944443 1.00 AGTR2 (0.50) AGTR2OXTRALDH1A1SMN1; SMN2MEN1
SCHEMBL4944440 1.00 AGTR2 (0.50) AGTR2OXTRALDH1A1SMN1; SMN2MEN1
SCHEMBL4942624 0.89 AGTR2 (0.46) AGTR2OXTRALDH1A1SMN1; SMN2MEN1
SCHEMBL4942629 0.89 AGTR2 (0.46) AGTR2OXTRALDH1A1SMN1; SMN2MEN1
SCHEMBL4936068 0.89 OXTR (0.56) AGTR2OXTRAGTR1AVPR1A
SCHEMBL4936062 0.89 OXTR (0.56) AGTR2OXTRAGTR1AVPR1A
SCHEMBL5744747 0.83 OXTR (0.65) OXTRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL4940289 0.83 OXTR (0.65) OXTRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL5744744 0.83 OXTR (0.65) OXTRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL4942106 0.80 OXTR (0.51) AGTR2OXTRALDH1A1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030171309-A1 Pharmaceutically active pyrrolidine derivatives as bax inhibitors MERCK SERONO SA (CH) 2003-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030171309-A1 Pharmaceutically active pyrrolidine derivatives as bax inhibitors SUCNR1, PYCR1, GLS AGTR2 2446/4885OXTR 189/4885ALDH1A1 3249/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.