SCHEMBL7219252

SCHEMBL7219252

CC1NC(C)(Cc2ccccc2)C(=O)O1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.39
CYP3A4 P08684 1/20 0.35
PARP1 P09874 1/20 0.35
MMP2 P08253 2/20 0.35
MMP9 P14780 2/20 0.35
MMP8 P22894 2/20 0.35
MMP13 P45452 2/20 0.35
TLR9 Q9NR96 1/20 0.34
CTSG P08311 1/20 0.34
PRTN3 P24158 1/20 0.34
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215883 0.85 ADAM17 (0.36) MAPTKMT2ATP53
SCHEMBL7213677 0.84 GRM2 (0.38) LMNAMEN1KMT2A
SCHEMBL7220659 0.81 NPSR1 (0.44) MMP2MMP9MMP8MMP13TLR9
SCHEMBL2520593 0.79 ALDH1A1 (0.39) ELANECYP3A4TLR9MEN1KMT2A
SCHEMBL11256573 0.71 ELANE (0.40) ELANECYP3A4MMP2MMP9MMP8
SCHEMBL29195204 0.71 ELANE (0.46) ELANECYP3A4MMP2MMP9MMP8
SCHEMBL576624 0.70 ELANE (0.39) ELANECYP3A4PARP1MMP2MMP9
SCHEMBL9413704 0.68 ELANE (0.37) ELANECYP3A4PARP1CTSGPRTN3
SCHEMBL7097777 0.67 ALDH1A1 (0.60) ELANECYP3A4MMP2MMP9MMP8
SCHEMBL15972776 0.67 ALDH1A1 (0.60) ELANECYP3A4MMP2MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6504046-B1 Cyclization of nitriles using acids, to form oxazolinone chemical intermediates such as 2-phenyl-4-isopropyl-4-methyl-1,3-oxazol-5-one, used as fungicides IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2003-01-07 US disclosed
EP-1092705-A1 PROCESS FOR THE PREPARATION OF AMIDES IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2001-04-18 EP disclosed
US-4680284-A RENNIN INHIBITORS, HYPOTENSIVE AGENTS ABBOTT LABORATORIES (US) 1987-07-14 US disclosed
EP-0189203-A2 Peptidylaminodiols ABBOTT LABORATORIES (US) 1986-07-30 EP disclosed