SCHEMBL7219255

SCHEMBL7219255

CC1=NC(C)(Cc2ccccc2)C(=O)O1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.40
BACE1 P56817 1/20 0.39
CTSG P08311 1/20 0.35
PRTN3 P24158 1/20 0.35
TSHR P16473 2/20 0.34
PIK3CD O00329 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
SORT1 Q99523 1/20 0.33
MMP2 P08253 2/20 0.33
MMP9 P14780 2/20 0.33
MMP8 P22894 2/20 0.33
MMP13 P45452 2/20 0.33
KCNQ2 O43526 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272506 1.00 ELANE (0.40) ELANEBACE1CTSGPRTN3TSHR
SCHEMBL7220662 0.83 NPSR1 (0.41) ALDH1A1MMP2MMP9MMP8MMP13
SCHEMBL11268643 0.82 ALDH1A1 (0.40) ELANEBACE1PIK3CDALDH1A1GAA
SCHEMBL19239774 0.81 RAB9A (0.36) ALDH1A1GAA
SCHEMBL508332 0.80 ELANE (0.36) ELANEBACE1CTSGPRTN3PIK3CD
SCHEMBL7662936 0.69 MMP2 (0.37) BACE1ALDH1A1MMP2MMP9CYP1A2
SCHEMBL6827479 0.67 BACE1 (0.43) BACE1MMP2MMP9CYP2C9
SCHEMBL16174713 0.67 ELANE (0.44) ELANECTSGPRTN3ALDH1A1GAA
SCHEMBL16174913 0.66 ELANE (0.51) ELANEBACE1CTSGPRTN3ALDH1A1
SCHEMBL11256573 0.66 ELANE (0.40) ELANEBACE1CTSGPRTN3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6504046-B1 Cyclization of nitriles using acids, to form oxazolinone chemical intermediates such as 2-phenyl-4-isopropyl-4-methyl-1,3-oxazol-5-one, used as fungicides IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2003-01-07 US disclosed
EP-1092705-A1 PROCESS FOR THE PREPARATION OF AMIDES IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2001-04-18 EP disclosed
US-4680284-A RENNIN INHIBITORS, HYPOTENSIVE AGENTS ABBOTT LABORATORIES (US) 1987-07-14 US disclosed
EP-0189203-A2 Peptidylaminodiols ABBOTT LABORATORIES (US) 1986-07-30 EP disclosed