SCHEMBL7220201

SCHEMBL7220201

Cc1cccnc1SC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 2/20 0.36
PLAU P00749 1/20 0.36
KDM4E B2RXH2 1/20 0.36
RAB9A P51151 1/20 0.36
CYP2A6 P11509 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.34
HSP90AA1 P07900 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
GAA P10253 2/20 0.33
LMNA P02545 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
METAP2 P50579 1/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27880031 0.82 NOS3 (0.42) NOS3NOS1NOS2ALDH1A1NPC1
SCHEMBL245135 0.78 NOS3 (0.50) NOS3NOS1NOS2ALDH1A1NPC1
SCHEMBL18059729 0.78 L3MBTL1 (0.36) ALDH1A1KDM4EL3MBTL1HSP90AA1MAPT
SCHEMBL7220195 0.78 L3MBTL1 (0.33) KDM4EL3MBTL1SMN1; SMN2SLC22A12
SCHEMBL5640712 0.76
SCHEMBL7615368 0.74
SCHEMBL245136 0.74
SCHEMBL27013272 0.74
SCHEMBL14218666 0.74
Ammonia Solution, Strong SCHEMBL1845719 0.74 NOS3 (0.46) NOS3NOS1NOS2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140309413-A1 METHODS OF STEREOSELECTIVE SYNTHESIS OF SUBSTITUTED NUCLEOSIDE ANALOGS VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-16 US disclosed
US-6503898-B1 Administering 4,7-dibenzyl-5,6-dihydroxy-N,N*-di(m-aminobenzyl)--1,3-diazepin-2-one or salt to treat human immunodeficiency virus infection BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-01-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140309413-A1 METHODS OF STEREOSELECTIVE SYNTHESIS OF SUBSTITUTED NUCLEOSIDE ANALOGS NUDT1, PAPSS1, NT5C3B NOS3 3595/4885NOS1 3968/4885NOS2 4104/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.