SCHEMBL7223531

SCHEMBL7223531

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2cccc(O)c2)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
CNR2 P34972 1/20 0.33
CNR1 P21554 1/20 0.33
POLB P06746 1/20 0.33
ESR1 P03372 1/20 0.32
ESRRG P62508 1/20 0.32
ESR2 Q92731 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
HTR3E A5X5Y0 3/20 0.32
HTR3B O95264 3/20 0.32
CHRNA7 P36544 3/20 0.32
HTR3A P46098 3/20 0.32
HTR3D Q70Z44 3/20 0.32
HTR3C Q8WXA8 3/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225045 0.89 SLC6A3 (0.41) SLC6A2SLC6A4SLC6A3ADRB1ADRB3
SCHEMBL7226014 0.89 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3POLBCHRNA7
SCHEMBL7231868 0.89 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3
SCHEMBL7231813 0.89 CHRNA7 (0.34) SLC6A2SLC6A4SLC6A3ADRB1ADRB3
SCHEMBL7225381 0.89 HTR3E (0.37) SLC6A2SLC6A4SLC6A3HTR3EHTR3B
SCHEMBL7233323 0.88 ESR1 (0.37) SLC6A2SLC6A4SLC6A3ESR1ESRRG
SCHEMBL7230406 0.87 PARP14 (0.38) NPC1
SCHEMBL7232389 0.87 NPC1 (0.36) SLC6A2SLC6A4SLC6A3HTR3EHTR3B
SCHEMBL7225098 0.87 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3ESRRGHTR3A
SCHEMBL7230191 0.87 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed