SCHEMBL7230406

SCHEMBL7230406

NC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 2/20 0.38
PARP10 Q53GL7 2/20 0.38
TNKS O95271 1/20 0.38
PARP15 Q460N3 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
NPC1 O15118 1/20 0.36
OPRK1 P41145 8/20 0.36
PKM P14618 1/20 0.35
PARP1 P09874 1/20 0.34
KCNH2 Q12809 8/20 0.34
OPRM1 P35372 6/20 0.34
FAAH O00519 1/20 0.34
TRPA1 O75762 1/20 0.34
EPHX2 P34913 1/20 0.34
FAAH2 Q6GMR7 1/20 0.34
MGLL Q99685 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232389 0.91 NPC1 (0.36) NPC1PKM
SCHEMBL7231813 0.89 CHRNA7 (0.34) KCNH2
SCHEMBL7224931 0.88 F2 (0.37) PARP14PARP10PARP15PARP2CHRNB2
SCHEMBL7223531 0.87 CHRNB4 (0.40) NPC1
SCHEMBL7231868 0.87 SLC6A2 (0.41) EPHX2
SCHEMBL7225045 0.87 SLC6A3 (0.41) EPHX2
SCHEMBL7226014 0.87 SLC6A2 (0.41) NPC1OPRM1OPRD1
SCHEMBL7225381 0.86 HTR3E (0.37) NPC1KCNH2
SCHEMBL7225098 0.86 SLC6A2 (0.44) KCNH2MGLL
SCHEMBL7234327 0.85 KMT2A (0.36) CHRNB2CHRNA4NPC1KCNH2FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed