SCHEMBL7224442

SCHEMBL7224442

O=C(Cl)CSc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.52
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
IDO1 P14902 1/20 0.49
MAPT P10636 8/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
POLB P06746 1/20 0.46
CRHBP P24387 1/20 0.46
CASP3 P42574 1/20 0.46
CRHR2 Q13324 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
CES1 P23141 1/20 0.46
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL877985 0.84 FFAR1 (0.57) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL11212940 0.82 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AIDO1MAPT
SCHEMBL11212945 0.82 SMN1; SMN2 (0.58) ALDH1A1MEN1KMT2AIDO1MAPT
SCHEMBL7223184 0.80 HSP90AA1 (0.57) ALDH1A1MEN1KMT2AMAPTCYP2C19
SCHEMBL7916730 0.79 ALDH1A1 (0.48) ALDH1A1MEN1KMT2AIDO1MAPT
SCHEMBL11876632 0.78 ALDH1A1 (0.58) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL5288477 0.78 ALDH1A1 (0.58) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL8030765 0.78 ALDH1A1 (0.48) ALDH1A1MEN1KMT2AIDO1MAPT
SCHEMBL10741564 0.77 IDO1 (0.54) ALDH1A1MEN1KMT2AIDO1MAPT
SCHEMBL7955282 0.77 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AIDO1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6552226-B1 Rapid; low temperature; one pot synthesis; reduced catalytic quantities of such as lewis acid and tertiary amine; entiomerically pure products THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-04-22 US disclosed
WO-2002026683-A1 TANDEM ACYL-CLAISEN REARRANGEMENT IN THE PREPARATION OF CHIRAL PRODUCTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2002-04-04 WO disclosed
US-6359174-B1 REACTING ALLYL REACTANT WITH ACID CHLORIDE IN PRESENCE OF LEWIS ACID CATALYST THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2002-03-19 US disclosed