SCHEMBL7226773

SCHEMBL7226773

Brc1cnc2nc(C3CCC3)ccn12

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA3 P34903 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224641 0.69 KDM4E (0.33) AKT1AKT2
SCHEMBL6221427 0.66 GABRA1 (0.34) GABRA1GABRG2GABRB3GABRA3
SCHEMBL5261894 0.66 GABRA1 (0.59) GABRA1GABRG2GABRB3GABRA3
SCHEMBL7224848 0.66 GABRG2 (0.43) AKT1AKT2GABRA1GABRG2GABRB3
SCHEMBL6217604 0.66 GABRA1 (0.34) GABRA1GABRG2GABRB3GABRA3
SCHEMBL6217979 0.66 GABRA1 (0.34) GABRA1GABRG2GABRB3GABRA3
SCHEMBL31579337 0.65 CNR2 (0.34) AKT1AKT2
SCHEMBL28822458 0.64 PIK3CD (0.34)
SCHEMBL6221519 0.64 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA3
SCHEMBL5771903 0.64 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6642229-B2 Treatment of adverse neurological conditions MERCK SHARP & DOHME LTD. 2003-11-04 US disclosed