SCHEMBL7230535

SCHEMBL7230535

C=C(O[Si](C)(C)C)c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.38
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP2C9 P11712 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NPC1 O15118 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MPO P05164 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2A6 P11509 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL347522 0.80 TSHR (0.37) NAPRTALDH1A1LMNASMN1; SMN2KMT2A
SCHEMBL19938127 0.78 ALDH1A1 (0.39) ALDH1A1LMNASMN1; SMN2KMT2AMEN1
SCHEMBL7237319 0.77 CES2 (0.38) ALDH1A1LMNASMN1; SMN2TP53NPC1
SCHEMBL29177284 0.77 CES2 (0.38) ALDH1A1LMNAKMT2AMEN1NPSR1
SCHEMBL7338642 0.77 CES2 (0.38) LMNASMN1; SMN2KMT2AMEN1NPC1
SCHEMBL8215216 0.75 MAPT (0.48) HSD17B10ALDH1A1LMNACYP2C19SMN1; SMN2
SCHEMBL8954661 0.75 MAPT (0.32)
SCHEMBL8459393 0.75 HPGD (0.50) NAPRTHSD17B10ALDH1A1SMN1; SMN2KMT2A
SCHEMBL8384037 0.74 PLK1 (0.40) HSD17B10ALDH1A1LMNACYP1A2SMN1; SMN2
SCHEMBL28971992 0.74 MAPT (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6503917-B1 Post-menopause, atherosclerosis, osteoporosis, and Alzheimer*s disease treatment WYETH, FIVE GIRALDA FARMS 2003-01-07 US disclosed
US-6384058-B1 COMPOUNDS AS ESTROGENS FOR TREATMENT OF DEFICIENCY AMERICAN HOME PRODUCTS CORPORATION 2002-05-07 US disclosed
US-6384060-B1 COMPOUNDS AS ESTROGENS FOR TREATMENT OF DEFICIENCY AMERICAN HOME PRODUCTS CORPORATION 2002-05-07 US disclosed
US-6384057-B1 COMPOUNDS AS ESTROGENS FOR TREATMENT OF DEFICIENCY AMERICAN HOME PRODUCTS CORPORATION 2002-05-07 US disclosed