SCHEMBL7230650

SCHEMBL7230650

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(-c2ccc(Cl)cc2Cl)o1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
CNR1 P21554 5/20 0.41
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ACKR3 P25106 3/20 0.36
SLC6A3 Q01959 3/20 0.36
SLC6A4 P31645 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232713 0.88 HDAC1 (0.48) NPC1RAB9ACNR1MEN1KMT2A
SCHEMBL7231985 0.86 HDAC1 (0.46) NPC1RAB9ACNR1L3MBTL1SLC6A3
SCHEMBL7232162 0.84 HDAC1 (0.50) NPC1RAB9AALDH1A1SMN1; SMN2HDAC1
SCHEMBL7231176 0.84 CA12 (0.39) SLC6A3SLC6A4HDAC1HDAC6
SCHEMBL7230828 0.83 SLC6A3 (0.41) NPC1RAB9ACNR1MEN1ALDH1A1
SCHEMBL7232072 0.83 HTT (0.48) NPC1RAB9AMEN1ALDH1A1HPGD
SCHEMBL7233040 0.82 ACKR3 (0.53) ACKR3
SCHEMBL7231983 0.82 SLC6A3 (0.37) NPC1RAB9ACNR1MEN1ALDH1A1
SCHEMBL7230561 0.82 ITGB2 (0.35) CNR1MEN1ALDH1A1HPGDKMT2A
SCHEMBL7225689 0.81 FAAH (0.43) NPC1RAB9AMEN1KMT2AACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed