SCHEMBL7232153

SCHEMBL7232153

O=[N+]([O-])c1c[c]cc([N+](=O)[O-])c1Cl

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 3/20 0.52
TDP1 Q9NUW8 6/20 0.47
TSHR P16473 4/20 0.47
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 3/20 0.47
ALOX15 P16050 2/20 0.47
HPGD P15428 1/20 0.47
HIF1A Q16665 1/20 0.47
TXNRD1 Q16881 1/20 0.47
TXNRD3 Q86VQ6 1/20 0.47
TXNRD2 Q9NNW7 1/20 0.47
GPR35 Q9HC97 2/20 0.43
MAPK1 P28482 1/20 0.40
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28866741 0.80 ALDH1A1 (0.49) VCAM1TDP1TSHRALDH1A1CYP3A4
SCHEMBL57836 0.77 TSHR (0.40) TDP1TSHRALDH1A1CYP3A4ALOX15
SCHEMBL7615798 0.75 TDP1 (0.40) VCAM1TDP1TSHRALDH1A1CYP3A4
SCHEMBL221622 0.75 TDP1 (0.56) TDP1TSHRALDH1A1CYP3A4GPR35
SCHEMBL3036771 0.75 GPR35 (0.56) TDP1ALDH1A1CYP3A4ALOX15HPGD
SCHEMBL19859 0.73 VCAM1 (0.46) VCAM1TDP1TSHRALDH1A1CYP3A4
SCHEMBL1460867 0.72 TDP1 (0.61) VCAM1TDP1TSHRALDH1A1CYP3A4
SCHEMBL9452603 0.72 TSHR (0.59) VCAM1TDP1TSHRALDH1A1CYP3A4
SCHEMBL29259432 0.72 VCAM1 (0.36) VCAM1TDP1TSHRALDH1A1CYP3A4
SCHEMBL27817013 0.72 VCAM1 (0.44) VCAM1TDP1TSHRALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112694473-A 7, 9-disubstituted berberine derivative and preparation method and application thereof 南京林业大学 2021-04-23 CN claimed
EP-0464736-B1 A process for producing 5-amino-4-halogeno-1H-pyrazole compounds FUJI PHOTO FILM CO LTD (JP) 1997-01-02 EP claimed
US-5122612-A PROCESS FOR PRODUCING 5-AMINO-4-HALOGENO-1H-PYRAZOLE COMPOUNDS FUJI PHOTO FILM CO., LTD. (JP) 1992-06-16 US claimed
EP-0464736-A1 A process for producing 5-amino-4-halogeno-1H-pyrazole compounds Fuji Photo Film Co., Ltd. (JP) 1992-01-08 EP claimed
CN-112694473-B 7, 9-disubstituted berberine structural analogue and preparation method and application thereof 南京林业大学 2022-09-20 CN disclosed
CN-112694473-A 7, 9-disubstituted berberine derivative and preparation method and application thereof 南京林业大学 2021-04-23 CN disclosed
US-6534518-B1 Phosphodiesterase inhibitors for respiratory system disorders ALTANA PHARMA AG (DE) 2003-03-18 US disclosed
EP-1163226-A1 POLYSUBSTITUTED 6-PHENYLPHENANTHRIDINES WITH PDE-IV INHIBITING ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2001-12-19 EP disclosed
WO-2000042018-A1 POLYSUBSTITUTED 6-PHENYLPHENANTHRIDINES WITH PDE-IV INHIBITING ACTIVITY BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-07-20 WO disclosed
EP-0464736-B1 A process for producing 5-amino-4-halogeno-1H-pyrazole compounds FUJI PHOTO FILM CO LTD (JP) 1997-01-02 EP disclosed
US-5122612-A PROCESS FOR PRODUCING 5-AMINO-4-HALOGENO-1H-PYRAZOLE COMPOUNDS FUJI PHOTO FILM CO., LTD. (JP) 1992-06-16 US disclosed
EP-0464736-A1 A process for producing 5-amino-4-halogeno-1H-pyrazole compounds Fuji Photo Film Co., Ltd. (JP) 1992-01-08 EP disclosed
EP-0051818-B1 PROCESS FOR THE PRODUCTION OF DISCHARGE-RESIST PRINTS ON TEXTILE MATERIALS CASSELLA Aktiengesellschaft (DE) 1985-09-04 EP disclosed
US-4398913-A ALKALINE PASTES CASSELLA AKTIENGESELLSCHAFT (DE) 1983-08-16 US disclosed
EP-0051818-A1 Process for the production of discharge-resist prints on textile materials CASSELLA Aktiengesellschaft (DE) 1982-05-19 EP disclosed