SCHEMBL28866741

SCHEMBL28866741

O=[N+]([O-])c1c[c]cc(C(F)(F)F)c1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
CYP3A4 P08684 2/20 0.49
ALOX15 P16050 2/20 0.49
TSHR P16473 2/20 0.49
HPGD P15428 1/20 0.49
HIF1A Q16665 1/20 0.49
TXNRD1 Q16881 1/20 0.49
TXNRD3 Q86VQ6 1/20 0.49
TXNRD2 Q9NNW7 1/20 0.49
VCAM1 P19320 1/20 0.37
EPAS1 Q99814 3/20 0.36
VEGFA P15692 1/20 0.35
PTPN5 P54829 1/20 0.35
GPR35 Q9HC97 1/20 0.34
ARNT P27540 1/20 0.34
AR P10275 6/20 0.33
SIRT6 Q8N6T7 1/20 0.33
CES2 O00748 1/20 0.33
ABCB11 O95342 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232153 0.80 VCAM1 (0.52) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL29190084 0.79 ALDH1A1 (0.49) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL2287677 0.76 NOTUM (0.33)
SCHEMBL29751617 0.73 TSHR (0.59) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL9175349 0.73 TDP1 (0.50) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL147979 0.73 KIF11 (0.41) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL317776 0.73 CYP3A4 (0.42) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL7745645 0.73 TSHR (0.59) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL10414958 0.71 CYP3A4 (0.79) ALDH1A1TDP1CYP3A4ALOX15TSHR
SCHEMBL1943291 0.71 ALDH1A1 (0.58) ALDH1A1TDP1CYP3A4ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601150-A Fused bicyclic RAF inhibitors and methods of use thereof 爵士制药爱尔兰有限公司 2023-08-15 CN disclosed
CN-108929329-A 2- azacyclo- -5- trifluoromethyl -8- nitro benzo (thio) pyrans -4- ketone compounds 中国医学科学院药物研究所 2018-12-04 CN disclosed