SCHEMBL7232158

SCHEMBL7232158

COc1ccccc1-c1ccc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 4/20 0.50
HSD17B10 Q99714 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
HPGD P15428 2/20 0.50
SLC9A1 P19634 1/20 0.45
RAB9A P51151 5/20 0.44
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 1/20 0.44
ATM Q13315 1/20 0.44
HTR3A P46098 2/20 0.43
CHRNA7 P36544 1/20 0.43
NPC1 O15118 4/20 0.42
LMNA P02545 2/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
ABCB1 P08183 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225355 0.90 ALDH1A1 (0.44) ALDH1A1KDM4EHSD17B10TDP1HPGD
SCHEMBL7232127 0.90 SLC9A1 (0.48) ALDH1A1KDM4EHSD17B10TDP1HPGD
SCHEMBL7222966 0.88 ALDH1A1 (0.53) ALDH1A1KDM4EHSD17B10TDP1HPGD
SCHEMBL7233102 0.87 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDSLC9A1RAB9A
SCHEMBL7226523 0.86 SMN1; SMN2 (0.42) ALDH1A1KDM4EHSD17B10HPGDRAB9A
SCHEMBL7234830 0.86 RAB9A (0.42) RAB9AMAPTSMN1; SMN2HTR3ANPC1
SCHEMBL7224300 0.85 RAB9A (0.40) ALDH1A1KDM4EHSD17B10TDP1HPGD
SCHEMBL7223501 0.85 RAB9A (0.40) ALDH1A1KDM4EHSD17B10TDP1HPGD
SCHEMBL7226764 0.85 RAB9A (0.53) ALDH1A1KDM4EHSD17B10TDP1HPGD
SCHEMBL7225840 0.85 RAB9A (0.41) ALDH1A1KDM4EHSD17B10HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed