SCHEMBL7225355

SCHEMBL7225355

COc1cccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)o2)c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
TSHR P16473 1/20 0.44
ATM Q13315 1/20 0.44
SLC6A3 Q01959 2/20 0.40
HPGD P15428 1/20 0.39
HTR3A P46098 2/20 0.39
CHRNA7 P36544 1/20 0.39
LMNA P02545 2/20 0.38
KDM1A O60341 1/20 0.38
S1PR2 O95136 1/20 0.38
S1PR4 O95977 1/20 0.38
S1PR3 Q99500 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232158 0.90 ALDH1A1 (0.50) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2
SCHEMBL7224676 0.88 SLC9A1 (0.45) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2
SCHEMBL7231044 0.86 RAB9A (0.37) KDM4EHSD17B10SMN1; SMN2RAB9ASLC6A3
SCHEMBL7072612 0.84 RAB9A (0.49) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2
Hydrochloric Acid SCHEMBL7070829 0.83 RAB9A (0.48) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2
SCHEMBL7222966 0.83 ALDH1A1 (0.53) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2
SCHEMBL7232127 0.82 SLC9A1 (0.48) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2
SCHEMBL7233102 0.82 ALDH1A1 (0.49) ALDH1A1KDM4ESMN1; SMN2MAPTRAB9A
SCHEMBL7226523 0.81 SMN1; SMN2 (0.42) ALDH1A1KDM4EHSD17B10SMN1; SMN2MAPT
SCHEMBL7232458 0.81 HTR4 (0.41) ALDH1A1KDM4EHSD17B10TDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed