SCHEMBL7248902

SCHEMBL7248902

Nc1cc(C(F)(F)F)c(-c2ccc(Cl)c(Cl)c2)cc1N1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.43
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
HTR3A P46098 1/20 0.39
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
HSD11B1 P28845 2/20 0.37
HTR7 P34969 3/20 0.36
TGFBR1 P36897 1/20 0.36
ACVR1 Q04771 1/20 0.36
NCF1 P14598 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
EPHX2 P34913 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6629232 0.78 ADRB1 (0.53) ADRB1HTR1AHTR3AHTR7NCF1
SCHEMBL7242525 0.78 ADRB1 (0.53) ADRB1HTR1AHTR3AHTR7NCF1
SCHEMBL7242984 0.71 HTT (0.49) ADRB1ADRB2HTR1AHTR3AHTR7
SCHEMBL2276545 0.67 ADRB2 (0.55) ADRB1ADRB2HTR1AHTR3ANCF1
SCHEMBL443520 0.67 HTR3A (0.51) ADRB1ADRB2HTR1AHTR3AHTR7
SCHEMBL6627622 0.67 ALDH1A1 (0.68) ADRB1ADRB2HTR1AHTR3ANCF1
SCHEMBL19403739 0.67 HTR3A (0.55) ADRB1ADRB2HTR1AHTR3AHTR7
SCHEMBL255333 0.67 ADRB1 (0.65) ADRB1ADRB2HTR1AHTR3AHTR7
SCHEMBL5252902 0.67 MAPT (0.52) ADRB1ADRB2HTR3ANCF1EPHX2
SCHEMBL7248900 0.66 ADRB1 (0.37) ADRB1HTR1AHTR3AAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030095958-A1 Inhibitors of bace VERTEX PHARMACEUTICALS INCORPORATED 2003-05-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030095958-A1 Inhibitors of bace BACE2, BACE1, APP ADRB1 3834/4885ADRB2 4466/4885HTR1A 4154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.