SCHEMBL7257015

SCHEMBL7257015

CC(C)(C)c1nc2[c]cccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 2/20 0.33
TXN P10599 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
PARP1 P09874 3/20 0.32
HDAC6 Q9UBN7 1/20 0.32
KCNH2 Q12809 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2901651 0.82 NPSR1 (0.53) L3MBTL1ALDH1A1SMN1; SMN2NPSR1PARP1
SCHEMBL3499660 0.76 NUDT1 (0.48) ALDH1A1
SCHEMBL211307 0.76 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2PARP1KDM4EGAA
SCHEMBL16095983 0.73
SCHEMBL5525401 0.72
SCHEMBL8470141 0.72
SCHEMBL7017594 0.71 KDM4E (0.32) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7021216 0.71 DDAH1 (0.53) L3MBTL1ALDH1A1SMN1; SMN2ADORA3ADORA2A
SCHEMBL7014749 0.71 LMNA (0.33) ALDH1A1GAAMAPT
SCHEMBL6197934 0.70 RAB9A (0.50) ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003053941-A2 BARBITURIC ACID DERIVATIVES AS INHIBITORS OF TNF-ALPHA CONVERTING ENZYME (TACE) AND/OR MATRIX METALLOPROTEINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-03 WO disclosed