SCHEMBL7257987

SCHEMBL7257987

COc1nc(N)c(Cl)cc1CC(=O)CC1CCN(CC(C)C)CC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.44
DRD4 P21917 2/20 0.44
KCNH2 Q12809 1/20 0.41
HTR4 Q13639 4/20 0.35
ACHE P22303 2/20 0.35
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254146 0.85 HTR4 (0.48) DRD2DRD4HTR4ACHEADRA2A
SCHEMBL7254103 0.81 HTR4 (0.42) DRD2DRD4HTR4ACHE
Hydrochloric Acid SCHEMBL8971647 0.81 DRD2 (0.52) DRD2DRD4HTR4ACHE
Hydrochloric Acid SCHEMBL7257861 0.81 HTR4 (0.41) DRD2DRD4HTR4ACHE
SCHEMBL6328978 0.78 HTR4 (0.54) HTR4ACHE
SCHEMBL7257990 0.76 KCNH2 (0.41) DRD2KCNH2HTR4ACHE
SCHEMBL7259161 0.72 KCNH2 (0.34) DRD2KCNH2
Hydrochloric Acid SCHEMBL8971855 0.72 DRD2 (0.50) DRD2DRD4HTR4ACHE
SCHEMBL8970802 0.70 HTR4 (0.61) DRD2DRD4HTR4ACHE
Hydrochloric Acid SCHEMBL8971667 0.69 HTR4 (0.60) DRD2DRD4HTR4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057688-A2 OXO OR OXY-PYRIDINE COMPOUNDS AS 5-HT4 RECEPTOR MODULATORS PFIZER JAPAN INC. (JP) 2003-07-17 WO claimed
WO-2003057688-A2 OXO OR OXY-PYRIDINE COMPOUNDS AS 5-HT4 RECEPTOR MODULATORS PFIZER JAPAN INC. (JP) 2003-07-17 WO disclosed