SCHEMBL7258750

SCHEMBL7258750

COc1ccc(N(N=O)c2ccc(OCc3cccnc3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.51
NFE2L2 Q16236 2/20 0.51
GRM2 Q14416 2/20 0.47
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.44
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
CYP19A1 P11511 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
MMP13 P45452 2/20 0.43
ACACB O00763 1/20 0.43
NR1D1 P20393 1/20 0.42
NR1H3 Q13133 1/20 0.42
GPR132 Q9UNW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7260721 0.90 NPC1 (0.53) GRM2HTTSMN1; SMN2NPC1MAPK1
SCHEMBL8361615 0.85 MAPK1 (0.56) HTTSMN1; SMN2NPC1GAAMAPK1
SCHEMBL7255278 0.84 NR4A2 (0.53) GRM2HTTSMN1; SMN2NPC1MAPK1
SCHEMBL6740488 0.81 NAMPT (0.54) HTTGAA
SCHEMBL6350923 0.78 GAA (0.79) HTTSMN1; SMN2NPC1GAAMAPK1
SCHEMBL7255986 0.78 CRHBP (0.54) NPC1GAAMAPK1HTR1ADRD2
SCHEMBL28048524 0.78 MAPK1 (0.64) HTTSMN1; SMN2MAPK1HTR1ADRD2
SCHEMBL7832381 0.74 CYP11B2 (0.57) NPC1MAPK1HTR1ADRD2CYP19A1
SCHEMBL29933468 0.74 CA1 (0.50) KEAP1NFE2L2SMN1; SMN2NPC1GAA
SCHEMBL7256123 0.73 RAB9A (0.74) HTTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003033467-A1 NITROSO DIPHENYLAMINE DERIVATIVES AS NITROGEN MONOXIDE GENERATING AGENTS MERCK PATENT GMBH (DE) 2003-04-24 WO disclosed