SCHEMBL7258766

SCHEMBL7258766

CC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@H](CO[Si](C)(C)C(C)(C)C)O[C@H]1n1c(-c2ccc(-c3ccccc3)cc2)nc2c(N)ncnc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.53
SIRT1 Q96EB6 1/20 0.53
GAPDH P04406 2/20 0.52
HSD17B10 Q99714 1/20 0.52
NADK O95544 1/20 0.51
TRPM2 O94759 5/20 0.49
SLC28A2 O43868 5/20 0.41
ADORA3 P0DMS8 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA2B P29275 2/20 0.41
ADORA1 P30542 2/20 0.41
PI4KA P42356 1/20 0.41
PI4K2B Q8TCG2 1/20 0.41
PI4K2A Q9BTU6 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
HSPA5 P11021 1/20 0.40
P2RX3 P56373 1/20 0.40
P2RX4 Q99571 1/20 0.40
P2RX2 Q9UBL9 1/20 0.40
GALR3 O60755 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254210 0.94 TRPM2 (0.47) SIRT2SIRT1GAPDHHSD17B10NADK
SCHEMBL1097330 0.88 SIRT2 (0.58) SIRT2SIRT1GAPDHHSD17B10NADK
SCHEMBL1097331 0.88 SIRT2 (0.58) SIRT2SIRT1GAPDHHSD17B10NADK
SCHEMBL1098546 0.86 GAPDH (0.55) SIRT2SIRT1GAPDHHSD17B10NADK
SCHEMBL7257500 0.84 ALDH1A1 (0.53) NADKADORA3ADORA2AADORA2BADORA1
SCHEMBL7257437 0.81 PRKAB2 (0.39) SIRT2SIRT1GAPDHHSD17B10TRPM2
SCHEMBL1097695 0.79 GAPDH (0.46) SIRT2SIRT1GAPDHHSD17B10NADK
SCHEMBL11417135 0.78 P2RX3 (0.52) GAPDHTRPM2SLC28A2ADORA3ADORA2A
SCHEMBL1098133 0.78 GAPDH (0.45) SIRT2SIRT1GAPDHHSD17B10NADK
SCHEMBL1097068 0.78 ALDH1A1 (0.47) SIRT2SIRT1GAPDHHSD17B10NADK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003051881-A1 SUBSTITUTED PURINE NUCLEOSIDE LIBRARIES AND COMPOUNDS BY SOLID-PHASE COMBINATORIAL STRATEGIES RIBAPHARM INC. (US) 2003-06-26 WO disclosed