SCHEMBL7258783

SCHEMBL7258783

C[C@H](O)[C@@H](CCOc1cccc(-c2ccc(Cl)nc2)c1)NC(=O)c1c[nH]cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.37
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
FAAH O00519 4/20 0.36
CHEK1 O14757 1/20 0.35
CHEK2 O96017 1/20 0.35
NAAA Q02083 1/20 0.35
SLC5A1 P13866 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GRM4 Q14833 1/20 0.34
ROCK1 Q13464 4/20 0.33
CNR1 P21554 1/20 0.33
MAP4K4 O95819 1/20 0.33
DYRK3 O43781 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7259490 0.91 CNR1 (0.39) ROCK2ACACBACACASLC5A1NPC1
SCHEMBL7263737 0.89 AVPR1B (0.41) SLC5A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL7258980 0.89 FAAH (0.42) ROCK2FAAHCHEK1CHEK2NPC1
SCHEMBL7264336 0.88 FAAH (0.34) ROCK2ACACBACACAFAAHCHEK1
SCHEMBL7259234 0.87 FFAR4 (0.41) ROCK2ACACBACACASLC5A1NPC1
SCHEMBL7263079 0.87 TP53 (0.46) ROCK2NPC1TP53RAB9ASMN1; SMN2
SCHEMBL7259217 0.86 SMN1; SMN2 (0.41) ROCK2ACACBACACANPC1TP53
SCHEMBL7259376 0.86 MRGPRX4 (0.39) ROCK2ACACBACACASLC5A1NPC1
SCHEMBL7263757 0.85 HDAC1 (0.40) SLC5A1
SCHEMBL7258877 0.82 SMN1; SMN2 (0.40) ROCK2NPC1TP53RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO claimed
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO disclosed