SCHEMBL7259376

SCHEMBL7259376

C[C@H](O)[C@@H](CCOc1cccc(-c2ccc(F)cc2)c1)NC(=O)c1c[nH]cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.39
ROCK1 Q13464 4/20 0.38
ROCK2 O75116 3/20 0.38
SCN9A Q15858 4/20 0.38
PDE2A O00408 1/20 0.38
NR4A2 P43354 3/20 0.38
DHODH Q02127 3/20 0.38
ACACB O00763 1/20 0.37
ACACA Q13085 1/20 0.37
HTR7 P34969 1/20 0.37
DYRK3 O43781 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CDK2 P24941 1/20 0.36
AKT2 P31751 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
IRAK1 P51617 1/20 0.36
PRKX P51817 1/20 0.36
CDK5 Q00535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7259490 0.92 CNR1 (0.39) ROCK1ROCK2ACACBACACADYRK3
SCHEMBL7259234 0.92 FFAR4 (0.41) ROCK1ROCK2ACACBACACADYRK3
SCHEMBL7259217 0.91 SMN1; SMN2 (0.41) ROCK1ROCK2ACACBACACANPC1
SCHEMBL7263079 0.90 TP53 (0.46) ROCK1ROCK2NPC1TP53RAB9A
SCHEMBL7263737 0.88 AVPR1B (0.41) SLC5A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL7258783 0.86 ROCK2 (0.37) ROCK1ROCK2ACACBACACADYRK3
SCHEMBL7258980 0.86 FAAH (0.42) ROCK1ROCK2NPC1TP53RAB9A
SCHEMBL7258877 0.84 SMN1; SMN2 (0.40) ROCK1ROCK2CDK2NPC1TP53
SCHEMBL7258741 0.84 HSD17B1 (0.38) ROCK1ACACBACACAPRKACAGSK3A
SCHEMBL7263757 0.84 HDAC1 (0.40) SLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO disclosed