SCHEMBL7259296

SCHEMBL7259296

CSc1ccc(-c2cc(=O)oc(N)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
XDH P47989 2/20 0.40
KDM4E B2RXH2 2/20 0.39
APP P05067 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTGS2 P35354 2/20 0.39
AR P10275 1/20 0.37
FBP1 P09467 1/20 0.36
MAPK13 O15264 1/20 0.36
GCGR P47871 1/20 0.36
MAPK12 P53778 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7261320 0.83 MEN1 (0.45) ADORA3ADORA2AADORA1KDM4EALDH1A1
SCHEMBL7261235 0.80 LTA4H (0.46) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL10827533 0.80 ADORA2A (0.52) ADORA2AADORA1XDHKDM4EALDH1A1
SCHEMBL4839060 0.76 KDM4E (0.48) ADORA3ADORA2AADORA2BADORA1KDM4E
SCHEMBL7022256 0.76 PGR (0.47) XDHGAAAR
SCHEMBL31298734 0.73 ADORA3 (0.44) ADORA3ADORA2AADORA2BADORA1XDH
SCHEMBL27195567 0.71 ADORA3 (0.54) ADORA3ADORA2AADORA2BADORA1XDH
SCHEMBL3452020 0.70 HSP90AA1 (0.64) ADORA3ADORA2AADORA2BADORA1KDM4E
SCHEMBL7702979 0.70 DYRK1A (0.46) ADORA3APP
SCHEMBL3451442 0.69 ADORA3 (0.44) ADORA3ADORA2AADORA2BADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084937-A2 PYRIMIDINEDIONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOLOGICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LIMITED (IN) 2003-10-16 WO disclosed