SCHEMBL7260713

SCHEMBL7260713

[O]Cc1cccc2[nH]c(Cl)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
PSMB8 P28062 1/20 0.37
ATP4A P20648 1/20 0.36
ATP4B P51164 1/20 0.36
CNR2 P34972 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
GRIN2B Q13224 1/20 0.35
MGAM O43451 3/20 0.34
GAA P10253 3/20 0.34
SI P14410 3/20 0.34
MGAM2 Q2M2H8 3/20 0.34
NUDT1 P36639 1/20 0.34
PARP1 P09874 5/20 0.34
ADORA1 P30542 2/20 0.33
MAOB P27338 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
GNRHR P30968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11398553 0.79 NPC1 (0.44) NPC1RAB9APSMB8ATP4AATP4B
SCHEMBL1128916 0.79 RAB9A (0.44) NPC1RAB9APSMB8ATP4AATP4B
SCHEMBL15111647 0.79 GAA (0.42) NPC1RAB9ACNR2GAAPARP1
SCHEMBL4191637 0.79 PARP1 (0.53) NPC1RAB9AATP4AATP4BCYP1A2
SCHEMBL9307952 0.78 NPC1 (0.46) NPC1RAB9ACYP1A2CYP2D6GRIN2B
SCHEMBL6829319 0.78 CHRM1 (0.46) NPC1RAB9ACNR2PARP1ALDH1A1
SCHEMBL629041 0.77 NPC1 (0.41) NPC1RAB9ACNR2CYP1A2MGAM
SCHEMBL3968950 0.76 DDAH1 (0.50) ATP4AATP4BGAAADORA1ADORA2A
SCHEMBL3973661 0.76 GRIN2B (0.36) NPC1RAB9ACYP1A2CYP2D6GRIN2B
SCHEMBL66295 0.75 PSMB8 (0.59) NPC1RAB9APSMB8MGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003053941-A2 BARBITURIC ACID DERIVATIVES AS INHIBITORS OF TNF-ALPHA CONVERTING ENZYME (TACE) AND/OR MATRIX METALLOPROTEINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-03 WO disclosed