SCHEMBL726261

SCHEMBL726261

NCc1cc(O)cc(CN)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.56
ABAT P80404 1/20 0.52
ACHE P22303 1/20 0.48
BACE1 P56817 2/20 0.41
TAAR1 Q96RJ0 3/20 0.41
DRD2 P14416 1/20 0.41
DRD1 P21728 1/20 0.41
LTA4H P09960 1/20 0.40
PTGS2 P35354 3/20 0.37
CYP3A4 P08684 1/20 0.37
LOXL2 Q9Y4K0 2/20 0.36
HRH3 Q9Y5N1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
SLC6A2 P23975 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTR3A P46098 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL632507 0.94 ENPP2 (0.56) ENPP2ABATACHEBACE1TAAR1
Hydrochloric Acid SCHEMBL3175518 0.91 ENPP2 (0.54) ENPP2ABATACHEBACE1TAAR1
SCHEMBL10666038 0.87 ABAT (0.48) ENPP2ABATACHEBACE1TAAR1
SCHEMBL20101128 0.84 ENPP2 (0.48) ENPP2ABATACHEBACE1TAAR1
SCHEMBL63392 0.83 LOXL2 (0.47) ENPP2ABATTAAR1LOXL2HRH3
SCHEMBL24264540 0.82 IDO1 (0.46) ENPP2ABATACHEBACE1TAAR1
SCHEMBL12524829 0.82 CA12 (0.55) ENPP2ABATACHETAAR1DRD2
SCHEMBL2451874 0.82 PNMT (0.46) ENPP2ABATACHETAAR1CYP3A4
Hydrochloric Acid SCHEMBL28226722 0.79 LOXL2 (0.44) ENPP2ABATTAAR1LOXL2HRH3
SCHEMBL11941632 0.77 CALM1 (0.59) ENPP2BACE1PTGS2CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119433983-A Preparation method of hydrophobic breathable fabric 普宁市福武纺织有限公司 2025-02-14 CN claimed
EP-2585539-B1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS RHODIA OPERATIONS (FR) 2016-11-02 EP claimed
US-9150692-B2 Polyamide composition RHODIA OPERATIONS (FR) 2015-10-06 US claimed
EP-2920229-A1 ALIPHATIC/SEMI-AROMATIC BLOCK COPOLYAMIDE Rhodia Operations (FR) 2015-09-23 EP claimed
US-9012544-B2 Polyamide composition for surface-mounted components RHODIA OPERATIONS (FR) 2015-04-21 US claimed
EP-2451861-B1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2014-11-05 EP claimed
WO-2014076120-A1 ALIPHATIC/SEMI-AROMATIC BLOCK COPOLYAMIDE RHODIA OPERATIONS (FR) 2014-05-22 WO claimed
US-20130153643-A1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS RHODIA OPERATIONS (FR) 2013-06-20 US claimed
US-20130115836-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2013-05-09 US claimed
EP-2585539-A1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS Rhodia Operations (FR) 2013-05-01 EP claimed
EP-2571925-A1 COMPOSITE POLYAMIDE ARTICLE Rhodia Operations S.A. (FR) 2013-03-27 EP claimed
US-20120238164-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2012-09-20 US claimed
US-20120177922-A1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2012-07-12 US claimed
EP-2451864-A1 COMPOSITE POLYAMIDE ARTICLE Rhodia Opérations (FR) 2012-05-16 EP claimed
EP-2451861-A1 POLYAMIDE COMPOSITION Rhodia Opérations (FR) 2012-05-16 EP claimed
WO-2011161082-A1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS RHODIA OPERATIONS (FR) 2011-12-29 WO claimed
WO-2011144592-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2011-11-24 WO claimed
WO-2011003785-A1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2011-01-13 WO claimed
WO-2011003787-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2011-01-13 WO claimed
CN-119433983-A Preparation method of hydrophobic breathable fabric 普宁市福武纺织有限公司 2025-02-14 CN disclosed
CN-119433983-A Preparation method of hydrophobic breathable fabric 普宁市福武纺织有限公司 2025-02-14 CN disclosed
WO-2024177097-A1 HYDROXYL GROUP-CONTAINING POLYAMIDE RESIN COMPOSITION, LAMINATE, PACKAGING MATERIAL, AND GAS BARRIER MATERIAL 東洋紡株式会社 2024-08-29 WO disclosed
EP-3237545-B1 POLYAMIDE MIXTURE HAVING IMPROVED FLUIDITY SPECIALTY OPERATIONS FRANCE (FR) 2024-02-28 EP disclosed
US-20210339487-A1 METHOD FOR THE CONTINUOUS PRODUCTION OF A COMPOSITE MATERIAL PROFILE SECTION FROM THERMOPLASTIC POLYMER HAVING HIGH FLUIDITY RHODIA OPERATIONS (FR) 2021-11-04 US disclosed
CN-107109054-B Polyamide mixtures with improved flowability 罗地亚经营管理公司 2021-08-17 CN disclosed
CN-106939126-B Polyamide composition for surface mounting parts 高性能聚酰胺有限公司 2021-01-12 CN disclosed
CN-107969122-B Composite profile, method for the production thereof and composite article 罗地亚经营管理公司 2020-11-06 CN disclosed
US-10723879-B2 Polyamide mixture having improved fluidity RHODIA OPERATIONS (FR) 2020-07-28 US disclosed
US-10584241-B2 Thermoplastic composition having high fluidity RHODIA OPERATIONS (FR) 2020-03-10 US disclosed
EP-3237544-B1 THERMOPLASTIC COMPOSITION HAVING HIGH FLUIDITY RHODIA OPERATIONS (FR) 2020-02-12 EP disclosed
EP-2512785-B1 METHOD FOR MANUFACTURING POLYAMIDE COMPOSITE ITEMS RHODIA OPERATIONS (FR) 2019-07-31 EP disclosed
EP-2920229-B1 ALIPHATIC/SEMI-AROMATIC BLOCK COPOLYAMIDE RHODIA OPERATIONS (FR) 2019-02-13 EP disclosed
US-20180257318-A1 METHOD FOR THE CONTINUOUS PRODUCTION OF A COMPOSITE MATERIAL PROFILE SECTION FROM THERMOPLASTIC POLYMER HAVING HIGH FLUIDITY RHODIA OPERATIONS (FR) 2018-09-13 US disclosed
US-20170342267-A1 THERMOPLASTIC COMPOSITION HAVING HIGH FLUIDITY RHODIA OPERATIONS (FR) 2017-11-30 US disclosed
US-20170342268-A1 POLYAMIDE MIXTURE HAVING IMPROVED FLUIDITY SPECIALTY OPERATIONS FRANCE (FR) 2017-11-30 US disclosed
EP-3237545-A1 POLYAMIDE MIXTURE HAVING IMPROVED FLUIDITY Rhodia Operations (FR) 2017-11-01 EP disclosed
EP-3237182-A1 METHOD FOR THE CONTINUOUS PRODUCTION OF A COMPOSITE MATERIAL PROFILE SECTION FROM THERMOPLASTIC POLYMER HAVING HIGH FLUIDITY Rhodia Operations (FR) 2017-11-01 EP disclosed
EP-3237544-A1 THERMOPLASTIC COMPOSITION HAVING HIGH FLUIDITY Rhodia Operations (FR) 2017-11-01 EP disclosed
US-9688823-B2 Aliphatic/semi-aromatic block copolyamide RHODIA OPERATIONS (FR) 2017-06-27 US disclosed
EP-2585539-B1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS RHODIA OPERATIONS (FR) 2016-11-02 EP disclosed
US-20160272767-A1 ALIPHATIC/SEMI-AROMATIC BLOCK COPOLYAMIDE SPECIALTY OPERATIONS FRANCE (FR) 2016-09-22 US disclosed
WO-2016102481-A1 THERMOPLASTIC COMPOSITION HAVING HIGH FLUIDITY RHODIA OPERATIONS (FR) 2016-06-30 WO disclosed
WO-2016102507-A1 POLYAMIDE MIXTURE HAVING IMPROVED FLUIDITY RHODIA OPERATIONS (FR) 2016-06-30 WO disclosed
US-9150692-B2 Polyamide composition RHODIA OPERATIONS (FR) 2015-10-06 US disclosed
EP-2920229-A1 ALIPHATIC/SEMI-AROMATIC BLOCK COPOLYAMIDE Rhodia Operations (FR) 2015-09-23 EP disclosed
US-9012544-B2 Polyamide composition for surface-mounted components RHODIA OPERATIONS (FR) 2015-04-21 US disclosed
EP-2451861-B1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2014-11-05 EP disclosed
WO-2014076120-A1 ALIPHATIC/SEMI-AROMATIC BLOCK COPOLYAMIDE RHODIA OPERATIONS (FR) 2014-05-22 WO disclosed
US-20130231335-A1 INHIBITORS OF POLO-LIKE KINASE ELAN PHARMACEUTICALS, INC. (US) 2013-09-05 US disclosed
US-20130153643-A1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS RHODIA OPERATIONS (FR) 2013-06-20 US disclosed
US-20130115836-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2013-05-09 US disclosed
EP-2585539-A1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS Rhodia Operations (FR) 2013-05-01 EP disclosed
EP-2571925-A1 COMPOSITE POLYAMIDE ARTICLE Rhodia Operations S.A. (FR) 2013-03-27 EP disclosed
EP-2512785-A1 METHOD FOR MANUFACTURING POLYAMIDE COMPOSITE ITEMS Rhodia Operations (FR) 2012-10-24 EP disclosed
US-20120238164-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2012-09-20 US disclosed
US-20120177922-A1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2012-07-12 US disclosed
EP-2451864-A1 COMPOSITE POLYAMIDE ARTICLE Rhodia Opérations (FR) 2012-05-16 EP disclosed
EP-2451861-A1 POLYAMIDE COMPOSITION Rhodia Opérations (FR) 2012-05-16 EP disclosed
WO-2011161082-A1 POLYAMIDE COMPOSITION FOR SURFACE-MOUNTED COMPONENTS RHODIA OPERATIONS (FR) 2011-12-29 WO disclosed
WO-2011144592-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2011-11-24 WO disclosed
WO-2011073198-A1 METHOD FOR MANUFACTURING POLYAMIDE COMPOSITE ITEMS RHODIA OPERATIONS (FR) 2011-06-23 WO disclosed
WO-2011003785-A1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2011-01-13 WO disclosed
WO-2011003785-A1 POLYAMIDE COMPOSITION RHODIA OPERATIONS (FR) 2011-01-13 WO disclosed
WO-2011003787-A1 COMPOSITE POLYAMIDE ARTICLE RHODIA OPERATIONS (FR) 2011-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130231335-A1 INHIBITORS OF POLO-LIKE KINASE POLK, PLK1, POLR2E ENPP2 2802/4885ABAT 3223/4885ACHE 1342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.