SCHEMBL7264698

SCHEMBL7264698

CCc1cc(I)cc2ccc(=O)[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.41
CA12 O43570 5/20 0.41
CA9 Q16790 5/20 0.41
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
F11 P03951 1/20 0.33
CA1 P00915 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA13 Q8N1Q1 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921146 0.77 DAO (0.41) DAOGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL29241812 0.74 CA12 (0.56) DAOCA12CA9GRIN2DGRIN3B
SCHEMBL8919065 0.74 CA12 (0.56) DAOCA12CA9GRIN2DGRIN3B
SCHEMBL7264685 0.74 GABRA1 (0.41) DAOCA12CA9F11CA1
SCHEMBL8918029 0.73 DAO (0.38) DAOCA12CA9ADRB2ADRB1
SCHEMBL8919183 0.73 CHEK1 (0.43) DAOCA12CA9CA1CA7
SCHEMBL8896840 0.69 CA12 (0.55) DAOCA12CA9GRIN2DGRIN3B
SCHEMBL17505173 0.68 GPR84 (0.47) ADRB2KDM4E
SCHEMBL8919040 0.67 PPARG (0.38) DAOPDE3BPDE3ARXFP1KDM4E
SCHEMBL8921004 0.67 CA12 (0.51) DAOCA12CA9CA1CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4710507-A Quinolone inotropic agents PFIZER INC. (US) 1987-12-01 US disclosed
CN-85100796-A The preparation method of qualone derivative 1986-10-01 CN disclosed
EP-0148623-A2 Quinolone inotropic agents Pfizer Limited (GB) 1985-07-17 EP disclosed