SCHEMBL7266284

SCHEMBL7266284

COC(C)NC(=O)c1ccc(-c2nc3cccc4c3n2CCC4=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.44
TP53 P04637 1/20 0.36
HTR3A P46098 1/20 0.35
CNR2 P34972 1/20 0.34
KCNH2 Q12809 2/20 0.34
GRM2 Q14416 2/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7261107 0.84 ROCK2 (0.48) PARP1
SCHEMBL7266288 0.83 NPC1 (0.47) PARP1TP53
SCHEMBL7260415 0.82 ROCK1 (0.43) PARP1
SCHEMBL7265103 0.79 NPC1 (0.46) PARP1TP53HTR3A
SCHEMBL7260381 0.79 NPC1 (0.46) PARP1TP53HTR3A
SCHEMBL7260372 0.78 MAPK14 (0.45) PARP1KCNH2GRM2
SCHEMBL7266685 0.77 NPSR1 (0.49)
SCHEMBL7261085 0.76 MMP13 (0.49) PARP1
SCHEMBL6199833 0.75 PARP1 (0.66) PARP1HTR3AKCNH2GRM2
SCHEMBL7266274 0.75 HPGD (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003103666-A2 NOVEL 4,5-DIHYDRO-IMIDAZO[4,5,1-IJ]QUINOLIN-6-ONES ALTANA PHARMA AG (DE) 2003-12-18 WO claimed
WO-2003103666-A2 NOVEL 4,5-DIHYDRO-IMIDAZO[4,5,1-IJ]QUINOLIN-6-ONES ALTANA PHARMA AG (DE) 2003-12-18 WO disclosed