SCHEMBL7266344

SCHEMBL7266344

C=CCc1cc[c]c2c1OCO2

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
ALOX15 P16050 1/20 0.40
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
POLB P06746 2/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623768 0.73 CYP3A4 (0.33) CYP3A4ALOX15CYP1A2MAPTPOLB
SCHEMBL5872023 0.72 NQO2 (0.30)
SCHEMBL4381961 0.68 AOC3 (0.32)
SCHEMBL1773996 0.64 GABRA1 (0.32) GABRA1GABRB2
SCHEMBL2946940 0.64 GABRA1 (0.35) GABRA1GABRB2
SCHEMBL5726097 0.63 CYP1A2 (0.36) CYP1A2
SCHEMBL7156166 0.63 GABRA1 (0.33) POLBGABRA1GABRB2
SCHEMBL723360 0.63 GABRA1 (0.33) CYP3A4CYP1A2MAPTGABRA1GABRB2
SCHEMBL7928568 0.63 GABRA1 (0.33) CYP3A4ALOX15ALDH1A1SMN1; SMN2GABRA1
SCHEMBL14552465 0.62 CYP3A4 (0.49) CYP3A4ALOX15CYP1A2MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003101381-A2 1,2 DIAMIDO CYCLOALKYL SODIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2003-12-11 WO disclosed