SCHEMBL7269133

SCHEMBL7269133

CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C(O)C(Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)CC

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.65
CTSL P07711 3/20 0.65
CTSS P25774 3/20 0.65
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
LMNA P02545 1/20 0.63
CTSD P07339 3/20 0.63
CASP3 P42574 2/20 0.57
REN P00797 1/20 0.56
CTSK P43235 3/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
RAB9A P51151 1/20 0.55
MME P08473 1/20 0.54
ECE1 P42892 1/20 0.54
TRPM8 Q7Z2W7 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448856 0.98 CTSB (0.65) CTSBCTSLCTSSMEN1KMT2A
SCHEMBL7277449 0.92 CTSL (0.57) CTSBCTSLCTSSMEN1KMT2A
SCHEMBL8769526 0.91 CTSL (0.63) CTSBCTSLCTSSMEN1KMT2A
SCHEMBL6449641 0.90 CTSD (0.76) CTSBCTSLCTSSCTSDCASP3
SCHEMBL6132144 0.90 CTSD (0.76) CTSBCTSLCTSSCTSDCASP3
SCHEMBL8769560 0.87 CTSD (0.65) CTSBCTSLCTSSMEN1KMT2A
Acetic Acid SCHEMBL7270658 0.87 CTSD (0.73) CTSBCTSLCTSSCTSDCASP3
SCHEMBL6446151 0.87 CTSD (0.76) CTSBCTSLCTSSCTSDCASP3
SCHEMBL6446780 0.87 CTSD (0.76) CTSBCTSLCTSSCTSDCASP3
SCHEMBL9232828 0.87 CTSD (0.76) CTSBCTSLCTSSCTSDCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed