SCHEMBL8769560

SCHEMBL8769560

CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)C(=O)NCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.65
CTSB P07858 3/20 0.61
CTSL P07711 3/20 0.61
CTSS P25774 3/20 0.61
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
LMNA P02545 1/20 0.59
PSMB1 P20618 1/20 0.58
CTSK P43235 2/20 0.53
TRPM8 Q7Z2W7 1/20 0.53
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
RAB9A P51151 1/20 0.52
CASP3 P42574 2/20 0.52
REN P00797 1/20 0.52
ANPEP P15144 1/20 0.50
BACE1 P56817 1/20 0.50
MME P08473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8769578 0.94 CTSD (0.59) CTSDCTSBCTSLCTSSMEN1
SCHEMBL8770005 0.91 CTSB (0.60) CTSDCTSBCTSLCTSSMEN1
SCHEMBL8769526 0.90 CTSL (0.63) CTSDCTSBCTSLCTSSMEN1
SCHEMBL8769497 0.89 REN (0.59) CTSDCTSBCTSLCTSSMEN1
SCHEMBL6448856 0.87 CTSB (0.65) CTSDCTSBCTSLCTSSMEN1
SCHEMBL7269133 0.87 CTSB (0.65) CTSDCTSBCTSLCTSSMEN1
SCHEMBL8770292 0.82 CTSB (0.61) CTSDCTSBCTSLCTSSMEN1
SCHEMBL7277449 0.80 CTSL (0.57) CTSDCTSBCTSLCTSSMEN1
SCHEMBL7425592 0.80 CTSD (0.67) CTSDCTSBCTSLCTSSCTSK
SCHEMBL8769553 0.80 BACE1 (0.49) CTSDKMT2APSMB1CYP3A4ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793673-A1 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR Takeda Chemical Industries, Ltd. (JP) 1997-09-10 EP disclosed
WO-1996016079-A2 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1996-05-30 WO disclosed