SCHEMBL7270150

SCHEMBL7270150

COC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CCCCCNC(=O)OCc1ccccc1)C(C)C)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
SIRT2 Q8IXJ6 3/20 0.49
SIRT1 Q96EB6 1/20 0.49
SIRT3 Q9NTG7 1/20 0.49
CAPN1 P07384 1/20 0.49
CAPN2 P17655 1/20 0.49
TGM2 P21980 1/20 0.49
PSMB5 P28074 1/20 0.48
FOLH1 Q04609 1/20 0.48
CPB1 P15086 1/20 0.47
CPB2 Q96IY4 1/20 0.47
CTSB P07858 1/20 0.47
CTSK P43235 1/20 0.47
CTSD P07339 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268430 0.93 HTT (0.52) HTTSIRT2SIRT1CAPN1CAPN2
SCHEMBL6443882 0.88 HTT (0.56) HTTSIRT2SIRT1SIRT3CAPN1
SCHEMBL6443877 0.88 HTT (0.56) HTTSIRT2SIRT1SIRT3CAPN1
SCHEMBL6447441 0.87 HTT (0.57) HTTSIRT2SIRT1CAPN1CAPN2
SCHEMBL6447440 0.87 HTT (0.57) HTTSIRT2SIRT1CAPN1CAPN2
SCHEMBL8539759 0.86 CTSD (0.57) PSMB5CTSD
SCHEMBL8534869 0.85 CTSD (0.58) HTTFOLH1CTSD
SCHEMBL9296228 0.84 CASP1 (0.54) CTSD
SCHEMBL30605359 0.83 HTT (0.48) HTTTGM2FOLH1CA2CA5A
SCHEMBL3210676 0.82 CTSB (0.60) CTSBCTSKCTSDCA2CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed