SCHEMBL7270440

SCHEMBL7270440

CC(C)[C@H](NC(=O)NCc1cccnc1)C(=O)NC(Cc1ccccc1)C(O)C(Cc1ccccc1)NC(=O)[C@@H](NC(=O)NCc1cccnc1)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
BACE1 P56817 6/20 0.52
CA2 P00918 1/20 0.52
CTSD P07339 3/20 0.52
LMNA P02545 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
PKM P14618 1/20 0.47
KMT2A Q03164 1/20 0.47
NAMPT P43490 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268683 0.92 CTSD (0.65) ALDH1A1BACE1CA2CTSD
SCHEMBL7269992 0.89 CTSD (0.61) BACE1CA2CTSDL3MBTL1
SCHEMBL7270439 0.84 CA2 (0.68) ALDH1A1BACE1CA2CTSD
SCHEMBL7269055 0.83 CA2 (0.52) BACE1CA2CTSDLMNANAMPT
SCHEMBL6446529 0.83 LMNA (0.56) BACE1CA2CTSDLMNAKMT2A
SCHEMBL7270066 0.83 CA2 (0.56) BACE1CA2CTSDLMNA
SCHEMBL7268971 0.82 CTSD (0.63) CA2CTSD
SCHEMBL6446176 0.82 ALDH1A1 (0.65) ALDH1A1L3MBTL1PKMKMT2A
SCHEMBL6446181 0.82 ALDH1A1 (0.65) ALDH1A1L3MBTL1PKMKMT2A
SCHEMBL7275770 0.82 CTSD (0.65) CA2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed