SCHEMBL7270838

SCHEMBL7270838

CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(N)=O)C(=O)NC(Cc1ccccc1)C(O)C(Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.70
CTSK P43235 10/20 0.62
CAPN1 P07384 2/20 0.61
CTSL P07711 5/20 0.58
REN P00797 1/20 0.57
CTSS P25774 2/20 0.56
CTSB P07858 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7277646 0.93 PSMB1 (0.62) PSMB1CTSKCAPN1REN
SCHEMBL7270223 0.92 PSMB1 (0.59) PSMB1CTSKCTSLRENCTSS
SCHEMBL6444976 0.90 CTSK (0.72) PSMB1CTSKCAPN1CTSLCTSS
SCHEMBL7267407 0.87 PSMB1 (0.70) PSMB1CTSKCAPN1CTSLCTSS
SCHEMBL27429302 0.87 PSMB1 (0.67) PSMB1CTSKCAPN1CTSLCTSS
SCHEMBL7279478 0.86 ADORA3 (0.56) PSMB1CTSKCTSLRENCTSS
SCHEMBL7270738 0.85 ADORA3 (0.63) PSMB1CTSKCTSLRENCTSS
SCHEMBL7418250 0.84 PSMB1 (0.61) PSMB1CTSKCAPN1CTSLREN
SCHEMBL7420596 0.84 PSMB1 (0.61) PSMB1CTSKCAPN1CTSLREN
SCHEMBL7412449 0.84 PSMB1 (0.61) PSMB1CTSKCAPN1CTSLREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed