SCHEMBL6444976

SCHEMBL6444976

CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C(O)C(O)C(Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.72
CTSL P07711 7/20 0.67
CAPN1 P07384 2/20 0.66
PSMB1 P20618 1/20 0.65
CTSS P25774 3/20 0.65
CTSB P07858 3/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8951282 0.91 CAPN1 (0.66) CTSKCTSLCAPN1PSMB1CTSS
SCHEMBL7270838 0.90 PSMB1 (0.70) CTSKCTSLCAPN1PSMB1CTSS
SCHEMBL6449605 0.89 TACR1 (0.69) CTSKCTSLCTSSCTSB
SCHEMBL7345360 0.87 CTSK (0.61) CTSKCTSLCAPN1PSMB1CTSS
SCHEMBL7345352 0.87 CTSK (0.61) CTSKCTSLCAPN1PSMB1CTSS
SCHEMBL6559243 0.86 CTSK (0.62) CTSKCTSLCAPN1PSMB1CTSS
SCHEMBL7327426 0.86 CAPN1 (0.78) CTSKCTSLCAPN1CTSSCTSB
SCHEMBL9828791 0.86 CAPN1 (0.78) CTSKCTSLCAPN1CTSSCTSB
SCHEMBL27809377 0.86 CAPN1 (0.78) CTSKCTSLCAPN1CTSSCTSB
SCHEMBL6446525 0.85 CTSD (0.60) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed