SCHEMBL7270960

SCHEMBL7270960

CC(Br)C1=Cc2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 3/20 0.52
CDC25A P30304 2/20 0.52
PTPN1 P18031 1/20 0.36
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
PTPRC P08575 1/20 0.30
CASP3 P42574 1/20 0.30
PLIN1 O60240 1/20 0.30
NR1I2 O75469 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GSR P00390 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
GAA P10253 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9471725 0.77 CDC25B (0.52) CDC25BCDC25APTPN1MEN1KMT2A
SCHEMBL3899596 0.71 CDC25A (0.60) CDC25BCDC25APTPN1
SCHEMBL31619928 0.70 CDC25B (0.89) CDC25BCDC25APTPN1MEN1KMT2A
SCHEMBL11828689 0.70 CDC25B (0.89) CDC25BCDC25APTPN1MEN1KMT2A
SCHEMBL2958225 0.67 LMNA (0.39) CDC25BCDC25APTPN1MEN1KMT2A
SCHEMBL7148148 0.64 HTR6 (0.35) CYP1A2CYP3A4CYP2D6CYP2C9MAOA
SCHEMBL6399287 0.64 CDC25B (0.47) CDC25BCDC25APTPN1MEN1KMT2A
SCHEMBL7270394 0.62
SCHEMBL826206 0.62
SCHEMBL1415318 0.61 P2RX7 (0.45) ALDH1A1LMNACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0457686-B1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1994-08-03 EP disclosed
US-5214055-A Analgesics, psychological disorders, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-05-25 US disclosed
US-5189045-A Antiserotonine agent ADIR ET COMPAGNIE (FR) 1993-02-23 US disclosed
EP-0457686-A1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-11-21 EP disclosed
US-5059674-A Cured arylcyclobutene ether spirodilactam SHELL OIL COMPANY (US) 1991-10-22 US disclosed
US-4968810-A Arylcyclobutene ethers SHELL OIL COMPANY (US) 1990-11-06 US disclosed