SCHEMBL7273155

SCHEMBL7273155

COc1cc(C(=O)N(C)CCN(C)C(=O)CC(c2ccc(F)cc2)c2ccc(F)cc2)cc(OC)c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.48
ALDH1A1 P00352 2/20 0.48
HPGD P15428 1/20 0.47
KCNH2 Q12809 3/20 0.42
TACR1 P25103 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KRAS P01116 1/20 0.40
ATM Q13315 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275717 0.85 TACR1 (0.47) SMN1; SMN2ALDH1A1HPGDKCNH2TACR1
Hydrochloric Acid SCHEMBL7267243 0.84 TACR1 (0.47) SMN1; SMN2ALDH1A1HPGDKCNH2TACR1
SCHEMBL7273027 0.81 CDK8 (0.47) SMN1; SMN2ALDH1A1L3MBTL1MAPK1KRAS
SCHEMBL9750661 0.79 SMN1; SMN2 (0.46) SMN1; SMN2ALDH1A1L3MBTL1KRASATM
SCHEMBL6596311 0.76 SMN1; SMN2 (0.40) SMN1; SMN2ALDH1A1KCNH2L3MBTL1NPSR1
SCHEMBL6596131 0.72 TUBB4A (0.40) SMN1; SMN2ALDH1A1KCNH2L3MBTL1KRAS
SCHEMBL9750679 0.71 SCN1A (0.49) ALDH1A1L3MBTL1MAPK1TUBB4ATUBB
Hydrochloric Acid SCHEMBL9750754 0.71 HPGD (0.55) SMN1; SMN2ALDH1A1HPGDKCNH2NPSR1
SCHEMBL7273776 0.71 L3MBTL1 (0.59) SMN1; SMN2ALDH1A1L3MBTL1MAPK1GAA
Hydrochloric Acid SCHEMBL9750696 0.70 SCN1A (0.48) SMN1; SMN2ALDH1A1L3MBTL1MAPK1TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293925-B1 COMPOUND ACTIVE IN CARDIOVASCULAR THERAPY SIMES, SOCIETA ITALIANA MEDICINALI E SINTETICI, S.P.A. (IT) 1991-10-16 EP disclosed
US-4988735-A Ethylene diamine active cardiovascular therapy SIMES (IT) 1991-01-29 US disclosed
EP-0293925-A2 Compound active in cardiovascular therapy SIMES, SOCIETA ITALIANA MEDICINALI E SINTETICI, S.P.A. (IT) 1988-12-07 EP disclosed