SCHEMBL9750661

SCHEMBL9750661

COc1cc(C(=O)N(C)CCN(C)C(=O)C=C(c2ccc(F)cc2)c2ccc(F)cc2)cc(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 1/20 0.46
KRAS P01116 1/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
TXNRD1 Q16881 1/20 0.41
TUBB4A P04350 6/20 0.41
TUBB P07437 6/20 0.41
TUBA3C P0DPH7 6/20 0.41
TUBA1B P68363 6/20 0.41
TUBA4A P68366 6/20 0.41
TUBB4B P68371 6/20 0.41
TUBB3 Q13509 6/20 0.41
TUBB2A Q13885 6/20 0.41
TUBB8 Q3ZCM7 6/20 0.41
TUBA3E Q6PEY2 6/20 0.41
TUBA1A Q71U36 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7267000 0.86 ALDH1A1 (0.44) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL7273027 0.80 CDK8 (0.47) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL7273155 0.79 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL8937380 0.76 KRAS (0.56) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL8937472 0.76 KRAS (0.56) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL8937377 0.76 KRAS (0.56) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL11115732 0.73 ACKR3 (0.45) SMN1; SMN2ALDH1A1L3MBTL1KDM4EMAPT
SCHEMBL8719068 0.72 PDE4A (0.49) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL8719072 0.72 PDE4A (0.49) SMN1; SMN2ALDH1A1KRASATML3MBTL1
SCHEMBL9750679 0.72 SCN1A (0.49) ALDH1A1L3MBTL1KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988735-A Ethylene diamine active cardiovascular therapy SIMES (IT) 1991-01-29 US disclosed