SCHEMBL727352

SCHEMBL727352

COc1cccc(OC)c1-c1cc(C(=O)N[C@H](c2nnn[nH]2)C2CCCCC2)nn1-c1cccc2ccccc12

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
APLNR P35414 8/20 0.49
PTGS2 P35354 1/20 0.42
NTSR1 P30989 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17114647 0.85 APLNR (0.56) APLNRNTSR1
SCHEMBL17114648 0.85 APLNR (0.56) APLNRNTSR1
SCHEMBL728944 0.85 NTSR1 (0.61) NTSR1
SCHEMBL727886 0.84 NTSR1 (0.50) APLNRPTGS2NTSR1
SCHEMBL17114580 0.78 PTGS2 (0.51) APLNRPTGS2NTSR1
SCHEMBL17114481 0.77 APLNR (0.44) APLNRPTGS2NTSR1
SCHEMBL8295919 0.75 NTSR1 (0.59) APLNRPTGS2NTSR1
SCHEMBL9083088 0.74 APLNR (0.52) APLNRNTSR1
SCHEMBL9086851 0.74 APLNR (0.52) APLNRNTSR1
SCHEMBL9084562 0.74 APLNR (0.51) APLNRNTSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011156557-A2 COMPOUNDS ACTIVE AT THE NEUROTENSIN RECEPTOR THOMAS JAMES B (US) 2011-12-15 WO disclosed