SCHEMBL7274253

SCHEMBL7274253

CCc1c(CO)ccc(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.45
AOC3 Q16853 1/20 0.44
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
CYP1A2 P05177 1/20 0.41
CHRM2 P08172 1/20 0.41
SLC6A4 P31645 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
KDM4E B2RXH2 3/20 0.40
TSHR P16473 1/20 0.40
APOBEC3A P31941 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
PTGS2 P35354 1/20 0.38
ALDH1A1 P00352 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30056339 0.89 AOC3 (0.46) AOC3PDE4APDE4BPDE4CPDE4D
SCHEMBL11300908 0.89 AOC3 (0.46) AOC3PDE4APDE4BPDE4CPDE4D
SCHEMBL7279487 0.86 AOC3 (0.45) SLC2A1AOC3PDE4APDE4BPDE4C
SCHEMBL1340134 0.84 AOC3 (0.53) AOC3PDE4APDE4BPDE4CPDE4D
SCHEMBL7273563 0.83 ALOX5 (0.47) SLC2A1AOC3SMN1; SMN2POLBKDM4E
Hydrochloric Acid SCHEMBL10648230 0.82 AOC3 (0.45) AOC3PDE4APDE4BPDE4CPDE4D
SCHEMBL11231888 0.81 TRPV1 (0.37) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL18475471 0.80 PTGS2 (0.46) SLC2A1AOC3SMN1; SMN2KDM4ETSHR
SCHEMBL9786067 0.80 HSD17B10 (0.51) SLC2A1PDE4DSMN1; SMN2KDM4ETSHR
SCHEMBL7274621 0.78 POLB (0.52) PDE4APDE4BPDE4CPDE4DSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed